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Discovery of AZD6642, an Inhibitor of 5-Lipoxygenase Activating Protein (FLAP) for the Treatment of Inflammatory Diseases
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Lemurell, Malin
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Ulander, Johan
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Dahlen, Anders
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Davidsson, Oejvind
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Emtenaes, Hans
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Broddefalk, Johan
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Swanson, Marianne
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Hovdal, Daniel
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Plowright, Alleyn T.
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Pettersen, Anna
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Ryden-Landergren, Marie
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Barlind, Jonas
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Llinas, Antonio
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Hersloef, Margareta
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Drmota, Tomas
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Sigfridsson, Kalle
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Moses, Sara
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Whatling, Carl
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JOURNAL OF MEDICINAL CHEMISTRY,
2015, 58 (02)
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Lemurell, Malin
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h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Ulander, Johan
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h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Winiwarter, Susanne
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Drug Safety & Metab, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Dahlen, Anders
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Davidsson, Oejvind
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Emtenaes, Hans
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Broddefalk, Johan
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Swanson, Marianne
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Hovdal, Daniel
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Plowright, Alleyn T.
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Pettersen, Anna
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Pharmaceut Dev, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Ryden-Landergren, Marie
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Resp Inflammat & Autoimmune Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Barlind, Jonas
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Llinas, Antonio
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h-index: 0
机构:
AstraZeneca, Resp Inflammat & Autoimmune Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Hersloef, Margareta
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Drmota, Tomas
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Resp Inflammat & Autoimmune Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Sigfridsson, Kalle
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Pharmaceut Dev, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Moses, Sara
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Drug Safety & Metab, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden

Whatling, Carl
论文数: 0 引用数: 0
h-index: 0
机构:
AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden AstraZeneca, Cardiovasc & Metab Dis iMed, S-43183 Molndal, Sweden
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Single-dose pharmacokinetics, pharmacodynamics and safety of AZD0837, a novel oral direct thrombin inhibitor, in young healthy male subjects
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INTERNATIONAL JOURNAL OF CLINICAL PHARMACOLOGY AND THERAPEUTICS,
2011, 49 (04)
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Johansson, S.
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h-index: 0
机构:
AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden

Cullberg, M.
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h-index: 0
机构:
AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden

Eriksson, U. G.
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h-index: 0
机构:
AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden

Elg, M.
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h-index: 0
机构:
AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden

Duner, K.
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h-index: 0
机构:
AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden

Jensen, E.
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h-index: 0
机构:
AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden

Wollbratt, M.
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h-index: 0
机构:
AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden

Wahlander, K.
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h-index: 0
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AstraZeneca R&D, S-43183 Molndal, Sweden AstraZeneca R&D, S-43183 Molndal, Sweden
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5-lipoxygenase-dependent biosynthesis of novel 20:4 n-3 metabolites with anti-inflammatory activity
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Gagnon, K. J.
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Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada

Lefort, N.
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h-index: 0
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Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada

Poirier, S. J.
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h-index: 0
机构:
Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada
Univ Laval, Inst Univ Cardiol & Pneumol Quebec, Ctr Rech, Quebec City, PQ, Canada Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada

Barnett, D. A.
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h-index: 0
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Atlantic Canc Res Inst, Moncton, NB, Canada Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada

Surette, M. E.
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h-index: 0
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Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada Univ Moncton, Dept Chim & Biochim, 18 Antonine Maillet Ave, Moncton, NB E1A 3E9, Canada
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Ezeamuzie, Charles, I
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Kuwait Univ, Fac Med, Dept Pharmacol & Toxicol, POB 24923, Safat 13110, Kuwait Kuwait Univ, Fac Med, Dept Pharmacol & Toxicol, POB 24923, Safat 13110, Kuwait

Rao, Muddanna S.
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h-index: 0
机构:
Kuwait Univ, Fac Med, Dept Anat, Safat, Kuwait Kuwait Univ, Fac Med, Dept Pharmacol & Toxicol, POB 24923, Safat 13110, Kuwait

El-Hashim, Ahmed Z.
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h-index: 0
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Kuwait Univ, Fac Pharm, Dept Pharmacol & Therapeut, Safat, Kuwait Kuwait Univ, Fac Med, Dept Pharmacol & Toxicol, POB 24923, Safat 13110, Kuwait

Philip, Elizabeth
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h-index: 0
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Kuwait Univ, Fac Med, Dept Pharmacol & Toxicol, POB 24923, Safat 13110, Kuwait Kuwait Univ, Fac Med, Dept Pharmacol & Toxicol, POB 24923, Safat 13110, Kuwait

Phillips, Oludotun A.
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Kuwait Univ, Fac Pharm, Dept Pharmaceut Chem, Safat, Kuwait Kuwait Univ, Fac Med, Dept Pharmacol & Toxicol, POB 24923, Safat 13110, Kuwait
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THE EFFECT OF MK-0591, A NOVEL 5-LIPOXYGENASE ACTIVATING PROTEIN INHIBITOR, ON LEUKOTRIENE BIOSYNTHESIS AND ALLERGEN-INDUCED AIRWAY RESPONSES IN ASTHMATIC SUBJECTS IN-VIVO
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JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY,
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DIAMANT, Z
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h-index: 0
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TIMMERS, MC
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h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA

VANDERVEEN, H
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h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA

FRIEDMAN, BS
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h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA

DESMET, M
论文数: 0 引用数: 0
h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA

DEPRE, M
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h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA

HILLIARD, D
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h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA

BEL, EH
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h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA

STERK, PJ
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h-index: 0
机构: MERCK RES LABS, RAHWAY, NJ USA
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Randomized, double-blinded, placebo-controlled phase I study of the pharmacokinetics, pharmacodynamics, and safety of KL130008, a novel oral JAK inhibitor, in healthy subjects
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Zhu, Xiaohong
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Fang, Fang
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Wang, Yongsheng
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Gong, Yimou
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Chen, Jing
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Gu, Liling
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EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES,
2022, 176

Li, Na
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h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Du, Shuangqing
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h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Wang, Ying
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h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Zhu, Xiaohong
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h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Shu, Shiqing
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h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Men, Yuchun
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h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

He, Miao
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h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Fang, Fang
论文数: 0 引用数: 0
h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Wang, Yongsheng
论文数: 0 引用数: 0
h-index: 0
机构:
Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Gong, Yimou
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h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Chen, Jing
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h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Gu, Liling
论文数: 0 引用数: 0
h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Cheng, Yezhe
论文数: 0 引用数: 0
h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

He, Qiang
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h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Lu, Huifang
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h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Niu, Yuanyuan
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h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Xu, Ying
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h-index: 0
机构:
Sichuan Kelun Biotech Biopharmaceut Co Ltd, Clin Res Ctr, 666 Xinhua Ave,Chengdu Cross Strait Sci & Technol, Chengdu 611100, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China

Feng, Ping
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h-index: 0
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Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China Sichuan Univ, West China Hosp, Clin Trial Ctr, Natl Med Prod Adm,Key Lab Clin Res & Evaluat Innov, Chengdu 610041, Sichuan, Peoples R China
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Bain, Gretchen
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Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

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Ziff, Jeannie
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Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

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h-index: 0
机构:
Amira Pharmaceut, Dept Drug Metab, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Baccei, Christopher
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Drug Metab, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Lee, Catherine
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Drug Metab, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Rong, Haojing
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Drug Metab, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Chapman, Charles
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Broadhead, Alex
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Lorrain, Dan
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Correa, Lucia
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Hutchinson, John H.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Evans, Jilly F.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA

Prasit, Peppi
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA Amira Pharmaceut, Dept Chem, San Diego, CA 92121 USA
[28]
Pharmacological Characterization of 3-[3-tert-Butylsulfanyl-1-[4-(6-methoxy-pyridin-3-yl)-benzyl]-5-(pyridin-2-ylmethoxy)-1H-indol-2-yl]-2,2-dimethyl-propionicAcid (AM103), a Novel Selective 5-Lipoxygenase-Activating Protein Inhibitor That Reduces Acute and Chronic Inflammation
[J].
Lorrain, Daniel S.
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Bain, Gretchen
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Correa, Lucia D.
;
Chapman, Charles
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Broadhead, Alex R.
;
Santini, Angelina M.
;
Prodanovich, Pat
;
Darlington, Janice V.
;
Hutchinson, John H.
;
King, Christopher
;
Lee, Catherine
;
Baccei, Christopher
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Li, Yiwei
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Arruda, Jeannie M.
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Evans, Jilly F.
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JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS,
2009, 331 (03)
:1042-1050

Lorrain, Daniel S.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Bain, Gretchen
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Correa, Lucia D.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Chapman, Charles
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Broadhead, Alex R.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Santini, Angelina M.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Prodanovich, Pat
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Darlington, Janice V.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Hutchinson, John H.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

King, Christopher
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Lee, Catherine
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Baccei, Christopher
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Li, Yiwei
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Arruda, Jeannie M.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA

Evans, Jilly F.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA Amira Pharmaceut, Dept Biol, San Diego, CA 92121 USA
[29]
Preclinical Pharmacokinetics and Acute Toxicity in Rats of 5-{[(2E)-3-Bromo-3-carboxyprop-2-enoyl]amino}-2-hydroxybenzoic Acid: A Novel 5-Aminosalicylic Acid Derivative with Potent Anti-Inflammatory Activity
[J].
Gutierrez-Sanchez, Mara
;
Romero-Castro, Aurelio
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Correa-Basurto, Jose
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Rosales-Hernandez, Martha Cecilia
;
Padilla-Martinez, Itzia Irene
;
Mendieta-Wejebe, Jessica Elena
.
MOLECULES,
2021, 26 (22)

Gutierrez-Sanchez, Mara
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico

Romero-Castro, Aurelio
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Quintana Roo, Div Ciencias Salud, Av Erick Paolo Martinez S-N,Esquina Av 4 Marzo, Chetmal 77039, Quintana Roo, Mexico Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico

Correa-Basurto, Jose
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad Invest, Lab Diseno & Desarrollo Nuevos Farmacos & Innovac, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico

Rosales-Hernandez, Martha Cecilia
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico

Padilla-Martinez, Itzia Irene
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Politecn Nacl, Unidad Prof Interdisciplinaria Biotecnol, Dept Ciencias Bas, Lab Quim Supramol & Nanociencias, Av Acueducto S-N,Colonia Barrio Laguna Ticoman, Mexico City 07340, DF, Mexico Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico

Mendieta-Wejebe, Jessica Elena
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico Inst Politecn Nacl, Escuela Super Med, Secc Estudios Posgrad & Invest, Lab Biofis & Biocatalisis, Plan San Luis & Salvador Diaz Miron S-N, Mexico City 11340, DF, Mexico
[30]
5-Lipoxygenase-activating protein inhibitors. Part 3: 3-{3-tert-Butylsulfanyl-1-[4-(5-methoxy-pyrimidin-2-yl)-benzyl]-5-(5-methylpyridin-2-ylmethoxy)-1H-indol-2-yl]-2,2-dimethyl-propionic acid (AM643)-A potent FLAP inhibitor suitable for topical administration
[J].
Stock, Nicholas
;
Baccei, Christopher
;
Bain, Gretchen
;
Chapman, Charles
;
Correa, Lucia
;
Darlington, Janice
;
King, Christopher
;
Lee, Catherine
;
Lorrain, Daniel S.
;
Prodanovich, Pat
;
Santini, Angelina
;
Schaab, Kevin
;
Evans, Jilly F.
;
Hutchinson, John H.
;
Prasit, Peppi
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2010, 20 (15)
:4598-4601

Stock, Nicholas
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Baccei, Christopher
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Bain, Gretchen
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Chapman, Charles
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Correa, Lucia
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Darlington, Janice
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

King, Christopher
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Lee, Catherine
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Lorrain, Daniel S.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Prodanovich, Pat
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Santini, Angelina
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Schaab, Kevin
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Evans, Jilly F.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Hutchinson, John H.
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA

Prasit, Peppi
论文数: 0 引用数: 0
h-index: 0
机构:
Amira Pharmaceut, San Diego, CA 92121 USA Amira Pharmaceut, San Diego, CA 92121 USA