A very short, efficient and inexpensive synthesis of the prodrug form of SC-54701A - A platelet aggregation inhibitor

被引：22

作者：

Cossy, J ^{[1
]}

Schmitt, A ^{[1
]}

Cinquin, C ^{[1
]}

Buisson, D ^{[1
]}

Belotti, D ^{[1
]}

机构：

[1] UNIV PARIS 05,CHIM & BIOCHIM PHARMACOL & TOXICOL LAB,CNRS,F-75270 PARIS 06,FRANCE

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1997年 / 7卷 / 13期

关键词：

D O I：

10.1016/S0960-894X(97)00293-X

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1699 / 1700

页数：2

共 16 条

[1] LOW-MOLECULAR-WEIGHT, NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONISTS [J].

ALIG, L ;

EDENHOFER, A ;

HADVARY, P ;

HURZELER, M ;

KNOPP, D ;

MULLER, M ;

STEINER, B ;

TRZECIAK, A ;

WELLER, T .

JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (23) :4393-4407

[2]

ANDRIEUX A, 1989, C INSERM, V174, P567

[3] SYNTHESIS OF OPTICALLY-ACTIVE T-BUTYL (3R,5S)-3,5-ISOPROPYLIDENEDIOXY-6-HEPTYNOATE THROUGH BAKERS-YEAST REDUCTION OF METHYL 3-OXO-4-PENTYNOATE [J].

ANSARI, MH ;

KUSUMOTO, T ;

HIYAMA, T .

TETRAHEDRON LETTERS, 1993, 34 (51) :8271-8274

[4]

BUISSON D, UNPUB

[5]

COSSY J, UNPUB

[6]

FABIANO E, 1987, SYNTHESIS-STUTTGART, P190

[7]

GOULD RJ, 1993, THROMB HAEMOSTASIS, V69, pA2

[8] NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONISTS .1. DISCOVERY AND DESIGN OF EXOSITE INHIBITORS [J].

HARTMAN, GD ;

EGBERTSON, MS ;

HALCZENKO, W ;

LASWELL, WL ;

DUGGAN, ME ;

SMITH, RL ;

NAYLOR, AM ;

MANNO, PD ;

LYNCH, RJ ;

ZHANG, GX ;

CHANG, CTC ;

GOULD, RJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (24) :4640-4642

[9] ETHYNYLSILANES .3. SYNTHESES OF SOME 2-ORGANOSILICON BICYCLO[2.2.1]HEPTADIENES AND BICYCLO[2.2.1]HEPT-2-ENES [J].

KRAIHANZEL, CS ;

LOSEE, ML .

JOURNAL OF ORGANIC CHEMISTRY, 1968, 33 (05) :1983-+

[10] THE USE OF DIETHYL AZODICARBOXYLATE AND TRIPHENYLPHOSPHINE IN SYNTHESIS AND TRANSFORMATION OF NATURAL-PRODUCTS [J].

MITSUNOBU, O .

SYNTHESIS-STUTTGART, 1981, (01) :1-28

← 1 2 →