Syntheses of New Carbanucleosides by Pericyclic Reactions

被引：17

作者：

Scagnelli, Luca ^{[1
]}

Memeo, Misal Giuseppe ^{[1
]}

Carosso, Serena ^{[1
]}

Bovio, Bruna ^{[1
]}

Quadrelli, Paolo ^{[1
]}

机构：

[1] Univ Pavia, Dept Chem, I-27100 Pavia, Italy

来源：

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | 2013年 / 2013卷 / 18期

关键词：

Antiviral agents; Carbanucleosides; Ene reaction; Cycloaddition; Nitrosocarbonyls; Nitrile oxides; CARBOCYCLIC NUCLEOSIDE ANALOGS; DIELS-ALDER REACTION; NITRILE OXIDES; MILD OXIDATION; ENE REACTIONS; BIOLOGICAL EVALUATION; ACYLNITROSO COMPOUNDS; HYDROXAMIC ACIDS; CONVENIENT ENTRY; 1ST SYNTHESIS;

D O I：

10.1002/ejoc.201300202

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of heterobase-functionalized cyclopentene derivatives as valuable substrate for the introduction of suitable substituents through pericyclic reactions is reported. The structures of ene and 1,3-dipolar adducts are discussed, and the primary antiviral activities of some adenine derivatives are reported.

引用

页码：3835 / 3846

页数：12

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