One-pot and two-step synthesis of novel carbonylthioureas and dicarbonyldithioureas derivatives

被引：7

作者：

Banaei, Alireza ^{[1
]}

Shiran, Jafar Abbasi ^{[1
]}

Saadat, Afshin ^{[2
]}

Ardabili, Farnaz Fazlalizadeh ^{[1
]}

McArdle, Patrick ^{[3
]}

机构：

[1] Payame Noor Univ, Dept Chem, Tehran, Iran

[2] Islamic Azad Univ, Germi Branch, Dept Chem, Gerrni, Iran

[3] NUI Galway, Dept Chem, Galway, Ireland

来源：

JOURNAL OF MOLECULAR STRUCTURE | 2015年 / 1099卷

关键词：

Carbonylthioureas; Dicarbonyldithioureas; Antibacterial activity; X-ray crystallography; ANTIBACTERIAL; SERIES; AGENTS; MOIETY;

D O I：

10.1016/j.molstruc.2015.06.074

中图分类号：

O64 [物理化学（理论化学）、化学物理学];

学科分类号：

070304 ; 081704 ;

摘要：

One-pot, two-step synthesis of several 1-cyclopropanecarbony1-3-(substituted phenyl)-thioureas and 1(phenylene-1,4-dione)-3,3'-(substituted phenyl)-dithioureas have been successfully prepared. The structures of the synthesized compounds were confirmed by elemental analysis, FT-IR spectroscopy and NMR. Also the crystal structure one of these compounds was determined by X-ray crystallography. All synthesized compounds were evaluated for antibacterial activity using Salmonella enterica (SE), Micrococcus luteus (ML), Bacillus subtilis (BS) and Pseudomonas aeruginosa (PS). (C) 2015 Elsevier B.V. All rights reserved.

引用

页码：427 / 431

页数：5

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