Molecular Basis for β-Glucosidase Inhibition by Ring-Modified Calystegine Analogues

被引：36

作者：

Aguilar, Matilde ^{[1
]}

Gloster, Tracey M. ^{[2
]}

Garcia-Moreno, M. Isabel ^{[1
]}

Mellet, Carmen Ortiz ^{[1
]}

Davies, Gideon J. ^{[2
]}

Llebaria, Amadeu ^{[4
]}

Casas, Josefina ^{[4
]}

Egido-Gabas, Meritxell ^{[4
]}

Fernandez, Jose M. Garcia ^{[3
]}

机构：

[1] Univ Seville, Fac Quim, Dept Quim Organ, Seville 41012, Spain

[2] York Struct Biol Lab, Dept Chem, York YO10 5YW, N Yorkshire, England

[3] Univ Seville, CSIC, Inst Invest Quim, Seville 41092, Spain

[4] Chem & Environm Res Inst Barcelona IIQBA CSIC, Res Unit Bioact Mol RUBAM, Barcelona 08034, Spain

来源：

CHEMBIOCHEM | 2008年 / 9卷 / 16期

基金：

英国生物技术与生命科学研究理事会;

关键词：

azasugars; calystegines; glucosidases; iminosugars; inhibitors;

D O I：

10.1002/cbic.200800451

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

[No abstract available]

引用

页码：2612 / 2618

页数：7

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