Lithium perchlorate assisted one-pot three-component aminoalkylation of electron-rich aromatic compounds

被引:71
作者
Saidi, MR [1 ]
Azizi, N [1 ]
Naimi-Jamal, MR [1 ]
机构
[1] Sharif Univ Technol, Dept Chem, Tehran, Iran
关键词
aminoalkylation; Mannich reaction; lithium perchlorate; electron-rich aromatic compounds;
D O I
10.1016/S0040-4039(01)01732-4
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A one-pot. three-component. Mannich reaction of electron-rich aromatic compounds with in situ prepared iminium salts in 5 M ethereal lithium perchlorate gives good yields of aminoalkylated products at room temperature. (C) 2001 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码:8111 / 8113
页数:3
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