Antivirals Targeting Influenza A Virus

被引:89
作者
Das, Kalyan [1 ]
机构
[1] Rutgers State Univ, Ctr Adv Biotechnol & Med, Dept Chem & Chem Biol, Piscataway, NJ 08854 USA
关键词
M2 PROTON CHANNELS; STRUCTURAL BASIS; RNA-POLYMERASE; ACTIVE-SITE; IN-VITRO; NEURAMINIDASE INHIBITORS; CRYSTAL-STRUCTURE; CAP-BINDING; ION-CHANNEL; AMINO-ACID;
D O I
10.1021/jm300455c
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:6263 / 6277
页数:15
相关论文
共 152 条
  • [71] Identification of influenza A nucleoprotein as an antiviral target
    Kao, Richard Y.
    Yang, Dan
    Lau, Lai-Shan
    Tsui, Wayne H. W.
    Hu, Lihong
    Dai, Jun
    Chan, Mei-Po
    Chan, Che-Man
    Wang, Pui
    Zheng, Bo-Jian
    Sun, Jian
    Huang, Jian-Dong
    Madar, Jason
    Chen, Guanhua
    Chen, Honglin
    Guan, Yi
    Yuen, Kwok-Yung
    [J]. NATURE BIOTECHNOLOGY, 2010, 28 (06) : 600 - U88
  • [72] Influenza neuraminidase inhibitors possessing a novel hydrophobic interaction in the enzyme active site: Design, synthesis, and structural analysis of carbocyclic sialic acid analogues with potent anti-influenza activity
    Kim, CU
    Lew, W
    Williams, MA
    Liu, HT
    Zhang, LJ
    Swaminathan, S
    Bischofberger, N
    Chen, MS
    Mendel, DB
    Tai, CY
    Laver, WG
    Stevens, RC
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1997, 119 (04) : 681 - 690
  • [73] T-705 (favipiravir) activity against lethal H5N1 influenza A viruses
    Kiso, Maki
    Takahashi, Kazumi
    Sakai-Tagawa, Yuko
    Shinya, Kyoko
    Sakabe, Saori
    Le, Quynh Mai
    Ozawa, Makoto
    Furuta, Yousuke
    Kawaoka, Yoshihiro
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2010, 107 (02) : 882 - 887
  • [74] GROWTH IMPAIRMENT RESULTING FROM EXPRESSION OF INFLUENZA-VIRUS M2 PROTEIN IN SACCHAROMYCES-CEREVISIAE - IDENTIFICATION OF A NOVEL INHIBITOR OF INFLUENZA-VIRUS
    KURTZ, S
    LUO, GX
    HAHNENBERGER, KM
    BROOKS, C
    GECHA, O
    INGALLS, K
    NUMATA, KI
    KRYSTAL, M
    [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1995, 39 (10) : 2204 - 2209
  • [75] SEQUENCES OF MESSENGER-RNAS DERIVED FROM GENOME RNA SEGMENT 7 OF INFLUENZA-VIRUS - COLINEAR AND INTERRUPTED MESSENGER-RNAS CODE FOR OVERLAPPING PROTEINS
    LAMB, RA
    LAI, CJ
    CHOPPIN, PW
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (07): : 4170 - 4174
  • [76] SITE-DIRECTED MUTATION OF THE ACTIVE-SITE OF INFLUENZA NEURAMINIDASE AND IMPLICATIONS FOR THE CATALYTIC MECHANISM
    LENTZ, MR
    WEBSTER, RG
    AIR, GM
    [J]. BIOCHEMISTRY, 1987, 26 (17) : 5351 - 5358
  • [77] The predominant mechanism by which ribavirin exerts its antiviral activity in vitro against flaviviruses and paramyxoviruses is mediated by inhibition of IMP dehydrogenase
    Leyssen, P
    Balzarini, J
    De Clercq, E
    Neyts, J
    [J]. JOURNAL OF VIROLOGY, 2005, 79 (03) : 1943 - 1947
  • [78] Crystal structure of the unique RNA-binding domain of the influenza virus NS1 protein
    Liu, JS
    Lynch, PA
    Chien, CY
    Montelione, GT
    Krug, RM
    Berman, HM
    [J]. NATURE STRUCTURAL BIOLOGY, 1997, 4 (11) : 896 - 899
  • [79] NUCLEAR TRANSPORT OF INFLUENZA-VIRUS RIBONUCLEOPROTEINS - THE VIRAL MATRIX PROTEIN (M1) PROMOTES EXPORT AND INHIBITS IMPORT
    MARTIN, K
    HELENIUS, A
    [J]. CELL, 1991, 67 (01) : 117 - 130
  • [80] The Effects of Influenza A Virus PB1-F2 Protein on Polymerase Activity Are Strain Specific and Do Not Impact Pathogenesis
    McAuley, Julie L.
    Zhang, Kelly
    McCullers, Jonathan A.
    [J]. JOURNAL OF VIROLOGY, 2010, 84 (01) : 558 - 564