Past, present and future of the Biginelli reaction: a critical perspective

被引:237
作者
Suresh [1 ]
Sandhu, Jagir S. [1 ]
机构
[1] Punjabi Univ, Dept Chem, Patiala 147002, Punjab, India
关键词
Biginelli reaction; multicomponent reactions; green process; ONE-POT SYNTHESIS; SOLVENT-FREE SYNTHESIS; MICROWAVE-ASSISTED SYNTHESIS; CALCIUM-CHANNEL BLOCKERS; HIGH-YIELDING PROTOCOL; CATALYZED EFFICIENT SYNTHESIS; POTASSIUM HYDROGEN SULFATE; SILICA SULFURIC-ACID; 3-COMPONENT CYCLOCONDENSATION REACTION; REUSABLE HETEROGENEOUS CATALYST;
D O I
10.3998/ark.5550190.0013.103
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
This review covers up to 2010 and some available references of 2011 of synthetic advances in the Biginelli reaction, including recent mechanistic advances, new building blocks, new pharmacological disclosures and asymmetric syntheses. Also present account is covering all aspects of the reaction whereas some of previous ones emphasized one aspect and others had passing reference.
引用
收藏
页码:66 / 133
页数:68
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