Structure activity relationships of tetrahydrocannabinol analogues on human cannabinoid receptors.

被引：85
作者：
Gareau, Y
Dufresne, C
Gallant, M
Rochette, C
Sawyer, N
Slipetz, DM
Tremblay, N
Weech, PK
Metters, KM
Labelle, M
机构：
[1] Merck Frosst Ctr. Therapeut. Res., Pointe-Claire-Dorval, Que. H9R 4P8
来源：
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1996年 / 6卷 / 02期
关键词：
D O I：
10.1016/0960-894X(95)00573-C
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A series of Delta(8)-tetrahydrocannabinol (THC) and biphenylic derivatives were prepared and their binding affinity for both human cannabinoid receptors hCB(1) and hCB(2) evaluated.
引用
收藏
页码：189 / 194
页数：6
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