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- [32] SAR study of bicyclo[4.1.0]heptanes as melanin-concentrating hormone receptor R1 antagonists: Taming hERGBIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (16) : 5369 - 5385Su, Jing论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAMcKittrick, Brian A.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USATang, Haiqun论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USABurnett, Duane A.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAClader, John W.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAGreenlee, William J.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAHawes, Brian E.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAO'Neill, Kim论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USASpar, Brian论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAWeig, Blair论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAKowalski, Timothy论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USASorota, Steve论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USALi, Cheng论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USALiu, Tongtong论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USA
- [33] Discovery of tetralin ureas as potent melanin concentrating hormone 1 receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (06) : 1718 - 1721Guo, Tao论文数: 0 引用数: 0 h-index: 0机构: Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USA Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USAGu, Huizhong论文数: 0 引用数: 0 h-index: 0机构: Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USA Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USAHobbs, Doug W.论文数: 0 引用数: 0 h-index: 0机构: Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USA Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USABusler, Dennis E.论文数: 0 引用数: 0 h-index: 0机构: Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USA Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USARokosz, Laura L.论文数: 0 引用数: 0 h-index: 0机构: Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USA Pharmacopeia Drug Discovery Inc, Princeton, NJ 08543 USA
- [34] Discovery of novel, orally available benzimidazoles as melanin concentrating hormone receptor 1 (MCHR1) antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (18) : 5443 - 5448Sasmal, Pradip K.论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaSasmal, Sanjita论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaRao, P. Tirumala论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaVenkatesham, B.论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaRoshaiah, M.论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaAbbineni, Chandrasekhar论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaKhanna, Ish论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaJadhav, Vikram P.论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaSuresh, J.论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaTalwar, Rashmi论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaMuzeeb, Syed论文数: 0 引用数: 0 h-index: 0机构: Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaReceveur, Jean-Marie论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma AS, DK-2970 Horsholm, Denmark Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaFrimurer, Thomas M.论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma AS, DK-2970 Horsholm, Denmark Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaRist, Oystein论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma AS, DK-2970 Horsholm, Denmark Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaElster, Lisbeth论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma AS, DK-2970 Horsholm, Denmark Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, IndiaHogberg, Thomas论文数: 0 引用数: 0 h-index: 0机构: 7TM Pharma AS, DK-2970 Horsholm, Denmark Dr Reddys Labs Ltd, Discovery Res, Hyderabad 500049, Andhra Pradesh, India
- [35] Discovery of melanin-concentrating hormone receptor R1 antagonists using high-throughput synthesisBIOORGANIC & MEDICINAL CHEMISTRY, 2005, 13 (05) : 1829 - 1836Su, J论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAMckittrick, BA论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USATang, HQ论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USACzarniecki, M论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAGreenlee, WJ论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAHawes, BE论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USAO'Neill, K论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Corp, Res Inst, Dept Chem Res, Kenilworth, NJ 07033 USA
- [36] Design and synthesis of orally efficacious benzimidazoles as melanin-concentrating hormone receptor 1 antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (14) : 3674 - 3678Wu, Wen-Lian论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USABurnett, Duane A.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USACaplen, Mary Ann论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USADomalski, Martin S.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USABennett, Chad论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USAGreenlee, William J.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USAHawes, Brian E.论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USAO'Neill, Kim论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USAWeig, Blair论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USAWeston, Daniel论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USASpar, Brian论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USAKowalski, Timothy论文数: 0 引用数: 0 h-index: 0机构: Schering Plough Res Inst, Kenilworth, NJ 07033 USA Schering Plough Res Inst, Kenilworth, NJ 07033 USA
- [37] SAR of biphenyl carboxamide ligands of the human melanin-concentrating hormone receptor 1 (MCH R1): Discovery of antagonist SB-568849BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (18) : 4865 - 4871Witty, David R.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandBateson, John H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandHervieu, Guillaume J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandJeffrey, Phillip论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandJohnson, Christopher N.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandMuir, Alison I.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandO'Hanlon, Peter J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandStemp, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandStevens, Alex J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandThewlis, Kevin M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandWilson, Shelagh论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, EnglandWinborn, Kim Y.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Harlow CM19 5AW, Essex, England GlaxoSmithKline, Harlow CM19 5AW, Essex, England
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