Copper-Catalyzed Synthesis of N-Heterocyclic Compounds

被引：97

作者：

Liu, Tao ^{[1
]}

Fu, Hua ^{[1
]}

机构：

[1] Tsinghua Univ, Dept Chem, Minist Educ, Key Lab Bioorgan Phosphorus Chem & Chem Biol, Beijing 100084, Peoples R China

来源：

SYNTHESIS-STUTTGART | 2012年 / 44卷 / 18期

基金：

中国国家自然科学基金;

关键词：

copper catalysis; N-heterocyclic compound; five-membered heterocycle; six-membered heterocycle; N-fused heterocycle; EFFICIENT SYNTHESIS; C-O; BOND FORMATION; COUPLING REACTION; CLICK CHEMISTRY; COPPER(I)-CATALYZED SYNTHESIS; BENZIMIDAZOLE DERIVATIVES; POLYSUBSTITUTED PYRROLES; REGIOSELECTIVE SYNTHESIS; SUBSTITUTED PYRROLES;

D O I：

10.1055/s-0032-1316763

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of N-heterocyclic compounds is an important direction because of their diverse biological functions. Recently, there has been remarkable progress in copper-catalyzed cross couplings with inexpensive, readily available, insensitive-to-air and low-toxicity copper catalysts. This review summarizes recent advances in the copper-catalyzed synthesis of N-heterocyclic compounds.

引用

页码：2805 / 2824

页数：20

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