Application of the aza-Wittig reaction for efficient synthesis of diversely substituted benzo[f]Chromeno[2,3-d]pyrimidine and benzo[f]chromeno[2,3-d][1,2,4]triazolopyrimidine derivatives

被引：1

作者：

Hassan, Mohamed ^{[1
]}

Barsy, Magda A. ^{[1
]}

El Rady, Eman A. ^{[1
]}

Al-Ayed, Abdullah Sulaiman ^{[2
]}

Frempong, Mona ^{[3
]}

Sadek, Kamal U. ^{[4
]}

机构：

[1] Aswan Univ, Fac Sci, Dept Chem, Aswan 81528, Egypt

[2] Qassim Univ, Coll Sci & Arts, Dept Chem, Ar Rass, Saudi Arabia

[3] Ctr Dis Control & Prevent, Atlanta, GA USA

[4] Minia Univ, Fac Sci, Chem Dept, Al Minya, Egypt

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2024年 / 61卷 / 04期

关键词：

ONE-POT SYNTHESIS; IN-VITRO; ANTITUMOR; DESIGN;

D O I：

10.1002/jhet.4784

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient synthesis of novel benzo[f]Chromeno[2,3-d]pyrimidine and unknown benzo[f]chromeno[2,3-d][1,2,4]triazolopyrimidine derivatives is described utilizing ethyl-2-amino-4-phenyl-4H-benzo[f]chromene-3-carboxyl-ate as precursor via aza-Wittig reaction. The process proved to be simple, high yielding, and efficient.

引用

页码：543 / 549

页数：7

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