Synthetic approaches to phosphonylpyridazines: an overview

被引：1

作者：

Abaid, Kmar ^{[1
]}

Touil, Soufiane ^{[1
]}

机构：

[1] Univ Carthage, Fac Sci Bizerte, Lab Heteroorgan Cpds & Nanostruct Mat LR18ES11, Jarzouna 7021, Tunisia

来源：

CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2023年 / 59卷 / 9-10期

关键词：

phosphonylpyridazines; pyridazines; cyclization; cycloaddition; phosphorylation; DIAZO-COMPOUNDS; AZIDES; ISOMERIZATION; CYCLOADDITION; SALTS;

D O I：

10.1007/s10593-023-03243-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Phosphonylpyridazines are an important class of compounds with promising applications in many fields, especially in medicinal chemistry. This review aims to describe the different strategies developed so far for the synthesis of phosphonylpyridazines, including phosphorylations on the pyridazine ring, as well as inter- and intramolecular cyclization reactions on functionalized phosphonates and phosphine oxides.

引用

收藏

页码：623 / 627

页数：5

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