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- [1] Discovery of a Bromodomain and Extra Terminal Domain (BET) Inhibitor with the Selectivity for the Second Bromodomain (BD2) and the Capacity for the Treatment of Inflammatory DiseasesJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (15) : 10824 - 10848Wang, Zhijie论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaYin, Li论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaXiong, Zhenghan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaHuang, Fei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaYang, Na论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaJiang, Fei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaLi, Huili论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaCui, Yong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaRen, Jiwei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaCheng, Zitian论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaJia, Kun论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaLu, Tao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaZhu, Jiapeng论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Med & Life Sci, State Key Lab Cultivat Base TCM Qual & Efficacy, Jiangsu Key Lab Pharmacol & Safety Evaluat Chinese, Nanjing 210023, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaHu, Qinghua论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaChen, Yadong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China
- [2] Discovery of a potent orally available pyrazolopyridone derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitorBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 109Hagihara, Shuichi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanIshizawa, Kouhei论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanSoga, Kana论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanHonjo, Takashi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanTakai, Shigeki论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanKawano, Yuko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanKikuchi, Manami论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanNishidate, Akiko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanMatsumoto, Fumi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanMurase, Mikako论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanHashimoto, Naohiro论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanSasaki, Chiduko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanMiyaguchi, Ikuko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanOkada, Okimasa论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanAkashi, Tomoya论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanNakayama, Shinji论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanOgasawara, Yuko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanEndo, Junichi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan
- [3] Discovery of a potent, orally available furopyridine derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitorBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 109Hagihara, Shuichi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanIshizawa, Kouhei论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanKikuchi, Manami论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanKawano, Yuko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanNishidate, Akiko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanMatsumoto, Fumi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanHashimoto, Naohiro论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanSasaki, Chiduko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanMiyaguchi, Ikuko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanOkada, Okimasa论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanAkashi, Tomoya论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanNakayama, Shinji论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanOgasawara, Yuko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, JapanEndo, Junichi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan Mitsubishi Tanabe Pharm Corp, Innovat Res Div, Sohyaku, 1000 Kamoshida Cho,Aoba Ku, Yokohama 2270033, Japan
- [4] Discovery of Tetrahydroquinoxalines as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the Second BromodomainJOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (10) : 4317 - 4334Law, Robert P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandAtkinson, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandBamborough, Paul论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandChung, Chun-wa论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandDemont, Emmanuel H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandGordon, Laurie J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Platform Technol & Sci, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandLindon, Matthew论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandPrinjha, Rab K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandWatson, Allan J. B.论文数: 0 引用数: 0 h-index: 0机构: Univ Strathclyde, Dept Pure & Appl Chem, WestCHEM, Thomas Graham Bldg,295 Cathedral St, Glasgow G1 1XL, Lanark, Scotland Univ St Andrews, Sch Chem, St Andrews KY16 9ST, Fife, Scotland GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, EnglandHirst, David J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Epigenet Discovery Performance Unit, Med Res Ctr, Stevenage SG1 2NY, Herts, England
- [5] A PET Imaging Probe Specifically Targeting the BD1 Bromodomain and Extra-Terminal DomainJOURNAL OF NUCLEAR MEDICINE, 2024, 65Wang, Yanli论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA USAWang, Changning论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA USA Massachusetts Gen Hosp, Boston, MA USAWang, Yongle论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Dept Radiol, Athinoula A Martinos Ctr Biomed Imaging, Boston, MA USA Harvard Med Sch, Boston, MA USA Massachusetts Gen Hosp, Boston, MA USA
- [6] Structure-Guided Design and Synthesis of Pyridinone-Based Selective Bromodomain and Extra-Terminal Domain (BET)-First Bromodomain (BD1) InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (04) : 2712 - 2731Li, Yangfeng论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA Chongqing Univ, Sch Pharmaceut Sci, Chongqing 401331, Peoples R China Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USAShen, Zhengnan论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USARatia, Kiira论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA Univ Illinois, Coll Pharm, Dept Biopharmaceut Sci, Chicago, IL 60612 USA Univ Illinois, Res Resources Ctr, Chicago, IL 60612 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USAZhao, Jiong论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Coll Pharm, Dept Biopharmaceut Sci, Chicago, IL 60612 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USAHuang, Fei论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USADubrovyskyii, Oleksii论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USAIndukuri, Divakar论文数: 0 引用数: 0 h-index: 0机构: Univ Arizona, Dept Pharmacol & Toxicol, Tucson, AZ 85721 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USAFu, Jiqiang论文数: 0 引用数: 0 h-index: 0机构: Univ Arizona, Dept Pharmacol & Toxicol, Tucson, AZ 85721 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USARamos, Omar Lozano论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, Res Resources Ctr, Chicago, IL 60612 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USAThatcher, Gregory R. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA Univ Illinois, Coll Pharm, Dept Biopharmaceut Sci, Chicago, IL 60612 USA Univ Arizona, Dept Pharmacol & Toxicol, Tucson, AZ 85721 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USAXiong, Rui论文数: 0 引用数: 0 h-index: 0机构: Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA Univ Illinois, Coll Pharm, Dept Biopharmaceut Sci, Chicago, IL 60612 USA Univ Arizona, Dept Pharmacol & Toxicol, Tucson, AZ 85721 USA Univ Illinois, UICtr Drug DiscoveryUIC, 833 S Wood St, Chicago, IL 60612 USA
- [7] GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) ProteinsJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (17) : 9045 - 9069Watson, Robert J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandBamborough, Paul论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Mol Discovery Res, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandBarnett, Heather论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Flexible Discovery Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandChung, Chun-wa论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Mol Discovery Res, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandDavis, Rob论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandGordon, Laurie论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Mol Discovery Res, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandGrandi, Paola论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Mol Discovery Res, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Cellzome GmbH, Mol Discovery Res, D-69117 Heidelberg, Germany GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandPetretich, Massimo论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Mol Discovery Res, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandPhillipou, Alex论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Mol Discovery Res, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandPrinjha, Rab K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandRioja, Inmaculada论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandSoden, Peter论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandWerner, Thilo论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Mol Discovery Res, Stevenage SG1 2NY, Herts, England GlaxoSmithKline, Cellzome GmbH, Mol Discovery Res, D-69117 Heidelberg, Germany GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, EnglandDemont, Emmanuel H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England GlaxoSmithKline Med Res Ctr, Epigenet Discovery Performance Unit, Stevenage SG1 2NY, Herts, England
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