Progress in Synthetic Trends Followed for the Development of 1,2,3-Triazole Derivatives: A Review

被引:7
作者
Masood, Mir Mohammad [1 ,2 ]
机构
[1] Govt Degree Coll Women Baramulla, Dept Chem, Baramulla, Jammu & Kashmir, India
[2] Govt Degree Coll Women Baramulla, Dept Chem, Baramulla 193101, Jammu & Kashmir, India
关键词
1,2,|3-Triazoles; Huisgen reactions; click chemistry; 1,3-dipolar cycloaddition; triazole synthesis; ONE-POT SYNTHESIS; AZIDE-ALKYNE CYCLOADDITION; ULTRASONIC-ASSISTED SYNTHESIS; CLICK CHEMISTRY; 1,4-DISUBSTITUTED 1,2,3-TRIAZOLES; COPPER-FREE; HIGHLY EFFICIENT; 1,3-DIPOLAR CYCLOADDITION; REGIOSELECTIVE SYNTHESIS; CATALYZED CYCLOADDITION;
D O I
10.1080/10406638.2023.2247119
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Since the beginning of click chemistry, 1,2,3-triazoles has been at the center of modern organic chemistry. This versatile framework has found broad applications in organic synthesis, drug discovery, chemical biology, polymer chemistry, supramolecular chemistry, bioconjugation, fluorescent imaging, and materials sciences. Due to tremendous use of 1,2,3-triazoles in chemistry, synthesis of this moiety from the easily available chemicals is desirable. This review covers different conventional and non-conventional approaches adopted for the synthesis of 1,2,3-triazole derivatives.
引用
收藏
页码:4273 / 4304
页数:32
相关论文
共 110 条
  • [1] Click Chemistry: 1,2,3-Triazoles as Pharmacophores
    Agalave, Sandip G.
    Maujan, Suleman R.
    Pore, Vandana S.
    [J]. CHEMISTRY-AN ASIAN JOURNAL, 2011, 6 (10) : 2696 - 2718
  • [2] A strain-promoted [3+2] azide-alkyne cycloaddition for covalent modification of blomolecules in living systems
    Agard, NJ
    Prescher, JA
    Bertozzi, CR
    [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2004, 126 (46) : 15046 - 15047
  • [3] Metal-free [3+2] cycloaddition of azides with Tf2C=CH2 for the regioselective preparation of elusive 4-(trifluoromethylsulfonyl)-1,2,3-triazoles
    Alcaide, Benito
    Almendros, Pedro
    Lazaro-Milla, Carlos
    [J]. CHEMICAL COMMUNICATIONS, 2015, 51 (32) : 6992 - 6995
  • [4] Synthesis and biological evaluation of novel 1,2,3-triazole derivatives as anti-tubercular agents
    Ali, Abdul Aziz
    Gogoi, Dhrubajyoti
    Chaliha, Amrita K.
    Buragohain, Alak K.
    Trivedi, Priyanka
    Saikia, Prakash J.
    Gehlot, Praveen S.
    Kumar, Arvind
    Chaturvedi, Vinita
    Sarma, Diganta
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 27 (16) : 3698 - 3703
  • [5] [Bmim]OH mediated Cu-catalyzed azide-alkyne cycloaddition reaction: A potential green route to 1,4-disubstituted 1,2,3-triazoles
    Ali, Abdul Aziz
    Konwar, Manashjyoti
    Chetia, Mitali
    Sarma, Diganta
    [J]. TETRAHEDRON LETTERS, 2016, 57 (50) : 5661 - 5665
  • [6] AgN(CN)2/DIPEA/H2O-EG: a highly efficient catalytic system for synthesis of 1,4-disubstituted-1,2,3 triazoles at room temperature
    Ali, Abdul Aziz
    Chetia, Mitali
    Saikia, Bishwajit
    Saikia, Prakash J.
    Sarma, Diganta
    [J]. TETRAHEDRON LETTERS, 2015, 56 (43) : 5892 - 5895
  • [7] Microwave versus conventional synthesis, anticancer, DNA binding and docking studies of some 1,2,3-triazoles carrying benzothiazole
    Aljuhani, Ateyatallah
    Almehmadi, Meshal A.
    Barnawi, Ibrahim O.
    Rezki, Nadjet
    Ali, Imran
    Messali, Mouslim
    Aouad, Mohamed Reda
    [J]. ARABIAN JOURNAL OF CHEMISTRY, 2021, 14 (03)
  • [8] Microwave-assisted benzyne-click chemistry: preparation of 1H-benzo[d][1,2,3]triazoles
    Ankati, Haribabu
    Biehl, Ed
    [J]. TETRAHEDRON LETTERS, 2009, 50 (32) : 4677 - 4682
  • [9] A microwave-assisted click chemistry synthesis of 1,4-disubstituted 1,2,3-triazoles via a copper(I)-catalyzed three-component reaction
    Appukkuttan, P
    Dehaen, W
    Fokin, VV
    Van der Eycken, E
    [J]. ORGANIC LETTERS, 2004, 6 (23) : 4223 - 4225
  • [10] Synthesis of 1,2-benzisoxazole tethered 1,2,3-triazoles that exhibit anticancer activity in acute myeloid leukemia cell lines by inhibiting histone deacetylases, and inducing p21 and tubulin acetylation
    Ashwini, Nanjundaswamy
    Garg, Manoj
    Mohan, Chakrabhavi Dhananjaya
    Fuchs, Julian E.
    Rangappa, Shobith
    Anusha, Sebastian
    Swaroop, Toreshettahally Ramesh
    Rakesh, Kodagahalli S.
    Kanojia, Deepika
    Madan, Vikas
    Bender, Andreas
    Koeffler, H. Phillip
    Basappa
    Rangappa, Kanchugarakoppal S.
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (18) : 6157 - 6165