共 45 条
HIPK1 Inhibition Protects against Pathological Cardiac Hypertrophy by Inhibiting the CREB-C/EBPβ Axis
被引:7
作者:

Bei, Yihua
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Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Zhu, Yujiao
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机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Wei, Meng
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机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Yin, Mingming
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Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Li, Lin
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机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Chen, Chen
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h-index: 0
机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Huang, Zhenzhen
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机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Liang, Xuchun
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机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Gao, Juan
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机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Yao, Jianhua
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机构:
Tongji Univ, Shanghai Peoples Hosp 10, Dept Cardiol, Sch Med, Shanghai 200072, Peoples R China
Shigatse Peoples Hosp, Dept Cardiol, Tibet 857000, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

van der Kraak, Petra H.
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机构:
Univ Utrecht, Univ Med Ctr Utrecht, Dept Pathol, NL-3584 CX Utrecht, Netherlands Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Vink, Aryan
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机构:
Univ Utrecht, Univ Med Ctr Utrecht, Dept Pathol, NL-3584 CX Utrecht, Netherlands Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Lei, Zhiyong
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机构:
Univ Utrecht, Univ Med Ctr Utrecht, Dept Cardiol, Lab Expt Cardiol, NL-3584 CX Utrecht, Netherlands
Univ Utrecht, Univ Med Ctr Utrecht, Div Lab, Cent Diag Lab Res, NL-3584 CX Utrecht, Netherlands Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Dai, Yuxiang
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机构:
Fudan Univ, Zhongshan Hosp, Shanghai Inst Cardiovasc Dis, Shanghai 200032, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Chen, Huihua
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机构:
Shanghai Univ Tradit Chinese Med, Sch Basic Med Sci, Shanghai 201203, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Liang, Yueyang
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Shanghai Univ Tradit Chinese Med, Sch Basic Med Sci, Shanghai 201203, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Sluijter, Joost P. G.
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机构:
Univ Utrecht, Univ Med Ctr Utrecht, Dept Cardiol, Lab Expt Cardiol, NL-3584 CX Utrecht, Netherlands
Univ Med Ctr Utrecht, UMC Utrecht Regenerat Med Ctr, NL-3508 GA Utrecht, Netherlands Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China

Xiao, Junjie
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h-index: 0
机构:
Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
机构:
[1] Shanghai Univ, Inst Geriatr, Affiliated Nantong Hosp, Peoples Hosp Nantong 6,Sch Med, Nantong 226011, Peoples R China
[2] Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Shanghai Engn Res Ctr Organ Repair,Sch Life Sci, Shanghai 200444, Peoples R China
[3] Tongji Univ, Shanghai Peoples Hosp 10, Dept Cardiol, Sch Med, Shanghai 200072, Peoples R China
[4] Shigatse Peoples Hosp, Dept Cardiol, Tibet 857000, Peoples R China
[5] Univ Utrecht, Univ Med Ctr Utrecht, Dept Pathol, NL-3584 CX Utrecht, Netherlands
[6] Univ Utrecht, Univ Med Ctr Utrecht, Dept Cardiol, Lab Expt Cardiol, NL-3584 CX Utrecht, Netherlands
[7] Univ Utrecht, Univ Med Ctr Utrecht, Div Lab, Cent Diag Lab Res, NL-3584 CX Utrecht, Netherlands
[8] Fudan Univ, Zhongshan Hosp, Shanghai Inst Cardiovasc Dis, Shanghai 200032, Peoples R China
[9] Shanghai Univ Tradit Chinese Med, Sch Basic Med Sci, Shanghai 201203, Peoples R China
[10] Univ Med Ctr Utrecht, UMC Utrecht Regenerat Med Ctr, NL-3508 GA Utrecht, Netherlands
基金:
欧洲研究理事会;
中国国家自然科学基金;
上海市自然科学基金;
关键词:
C/EBP beta;
cardiomyocytes;
CREB;
HIPK1;
pathological hypertrophy;
ACTIVATION;
GROWTH;
GENE;
LOCALIZATION;
REGULATOR;
PATHWAY;
ROLES;
D O I:
10.1002/advs.202300585
中图分类号:
O6 [化学];
学科分类号:
0703 ;
摘要:
Inhibition of pathological cardiac hypertrophy is recognized as an important therapeutic strategy for heart failure, although effective targets are still lacking in clinical practice. Homeodomain interacting protein kinase 1 (HIPK1) is a conserved serine/threonine kinase that can respond to different stress signals, however, whether and how HIPK1 regulates myocardial function is not reported. Here, it is observed that HIPK1 is increased during pathological cardiac hypertrophy. Both genetic ablation and gene therapy targeting HIPK1 are protective against pathological hypertrophy and heart failure in vivo. Hypertrophic stress-induced HIPK1 is present in the nucleus of cardiomyocytes, while HIPK1 inhibition prevents phenylephrine-induced cardiomyocyte hypertrophy through inhibiting cAMP-response element binding protein (CREB) phosphorylation at Ser271 and inactivating CCAAT/enhancer-binding protein.. (C/EBP ss)-mediated transcription of pathological response genes. Inhibition of HIPK1 and CREB forms a synergistic pathway in preventing pathological cardiac hypertrophy. In conclusion, HIPK1 inhibition may serve as a promising novel therapeutic strategy to attenuate pathological cardiac hypertrophy and heart failure.
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页数:15
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h-index: 0
机构: HELIOS Klin, Franz Volhard Clin, Berlin, Germany
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Long Noncoding RNA Cardiac Physiological Hypertrophy-Associated Regulator Induces Cardiac Physiological Hypertrophy and Promotes Functional Recovery After Myocardial Ischemia-Reperfusion Injury
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CIRCULATION,
2021, 144 (04)
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Gao, Rongrong
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h-index: 0
机构:
Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Wang, Lijun
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h-index: 0
机构:
Shanghai Univ, Shanghai Engn Res Ctr Organ Repair, Sch Med, Shanghai, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Sch Life Sci, 333 Nan Chen Rd, Shanghai 200444, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Bei, Yihua
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h-index: 0
机构:
Shanghai Univ, Shanghai Engn Res Ctr Organ Repair, Sch Med, Shanghai, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Sch Life Sci, 333 Nan Chen Rd, Shanghai 200444, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Wu, Xiaodong
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h-index: 0
机构:
Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Wang, Jiaqi
论文数: 0 引用数: 0
h-index: 0
机构:
Shanghai Univ, Shanghai Engn Res Ctr Organ Repair, Sch Med, Shanghai, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Sch Life Sci, 333 Nan Chen Rd, Shanghai 200444, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Zhou, Qiulian
论文数: 0 引用数: 0
h-index: 0
机构:
Shanghai Univ, Shanghai Engn Res Ctr Organ Repair, Sch Med, Shanghai, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Sch Life Sci, 333 Nan Chen Rd, Shanghai 200444, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Tao, Lichan
论文数: 0 引用数: 0
h-index: 0
机构:
Soochow Univ, Affiliated Hosp 3, Dept Cardiol, Changzhou, Jiangsu, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Das, Saumya
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h-index: 0
机构:
Massachusetts Gen Hosp, Cardiovasc Div, Boston, MA 02114 USA
Harvard Med Sch, Boston, MA 02115 USA Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Li, Xinli
论文数: 0 引用数: 0
h-index: 0
机构:
Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China

Xiao, Junjie
论文数: 0 引用数: 0
h-index: 0
机构:
Shanghai Univ, Shanghai Engn Res Ctr Organ Repair, Sch Med, Shanghai, Peoples R China
Shanghai Univ, Cardiac Regenerat & Ageing Lab, Inst Cardiovasc Sci, Sch Life Sci, 333 Nan Chen Rd, Shanghai 200444, Peoples R China Nanjing Med Univ, Affiliated Hosp 1, Dept Cardiol, 300 Guangzhou Rd, Nanjing 210029, Jiangsu, Peoples R China
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Cardiomyocyte Homeodomain-Interacting Protein Kinase 2 Maintains Basal Cardiac Function via Extracellular Signal-Regulated Kinase Signaling
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Guo, Yuanjun
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Willette, Robert N.
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Barnett, Joey V.
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Knollmann, Bjorn C.
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Force, Thomas
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Lal, Hind
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CIRCULATION,
2019, 140 (22)
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Guo, Yuanjun
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA
Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Sui, Jennifer Y.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Kim, Kyungsoo
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Clin Pharmacol, Nashville, TN USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Zhang, Zhentao
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA
Vanderbilt Univ, Dept Cell & Dev Biol, 221 Kirkland Hall, Nashville, TN 37235 USA
Vanderbilt Univ, Vanderbilt Ctr Stem Cell Biol, 221 Kirkland Hall, Nashville, TN 37235 USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Qu, Xiaoyan A.
论文数: 0 引用数: 0
h-index: 0
机构:
PAREXEL Int, Res Triangle Pk, NC USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Nam, Young-Jae
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA
Vanderbilt Univ, Dept Cell & Dev Biol, 221 Kirkland Hall, Nashville, TN 37235 USA
Vanderbilt Univ, Vanderbilt Ctr Stem Cell Biol, 221 Kirkland Hall, Nashville, TN 37235 USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Willette, Robert N.
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Metab Pathways & Cardiovasc Therapeut Area, Heart Failure Discovery Performance Unit, King Of Prussia, PA USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Barnett, Joey V.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Knollmann, Bjorn C.
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Clin Pharmacol, Nashville, TN USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Force, Thomas
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA

Lal, Hind
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA
Univ Alabama Birmingham, Div Cardiovasc Dis, 1720 2nd Ave South, Birmingham, AL 35294 USA Vanderbilt Univ, Med Ctr, Div Cardiovasc Med, Nashville, TN USA