Synthesis of benzothiazoles and biologically active derivatives from 2-aminothiophenol- REVIEW-

被引：1

作者：

Al-Mutairi, Aamal A. ^{[1
,2
]}

机构：

[1] Fac Sci, Chem Dept, Riyadh, Saudi Arabia

[2] Imam Mohammad Ibn Saud Islamic Univ IMSIU, POB 90950, Riyadh 11623, Saudi Arabia

来源：

EGYPTIAN JOURNAL OF CHEMISTRY | 2023年 / 66卷 / 13期

关键词：

Benzothiazole; 2-aminothiophenol; Antimicrobial; Anticancer; Biological applications; EFFICIENT SYNTHESIS; MANNICH-BASES; IN-SILICO; BENZIMIDAZOLES; DESIGN; BENZOXAZOLES; DOCKING; SEARCH; ADME; ACID;

D O I：

10.21608/EJCHEM.2023.195175.7630

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

In the new millennium, benzothiazole derivatives have attracted great interest in medicinal chemistry due to their pharmacological and biological properties. Benzothiazole nucleus possesses diverse biological properties such as antimicrobial, anticancer, antifungal, anthelmintic, antidiabetic and anticonvulsant activities. In this review, we expose the common procedures to synthesize benzothiazole and its derivatives, which comprise various biological activities.

引用

页码：923 / 937

页数：15

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