Efficacy and Safety of Poziotinib in HER2 Exon 20 Insertion NSCLC Patients who Received at Least 2 Previous Systemic Therapies

被引:0
|
作者
Le, X. [1 ]
Prelaj, A. [2 ]
Baik, C. [3 ]
Tchekmedyian, N. [4 ]
Leu, S. [5 ]
Bhat, G. [5 ]
Heymach, J. V. [1 ]
Cornelissen, R. [6 ]
机构
[1] MD Anderson Canc Ctr, Houston, TX USA
[2] Ist Nazl Tumori Milano Fdn IRCCS, Milan, Italy
[3] Seattle Canc Ctr Alliance, Seattle, WA USA
[4] City Hope Natl Med Ctr, Irvine, CA USA
[5] Spectrum Pharmaceut, Irvine, CA USA
[6] Erasmus MC Canc Inst, Rotterdam, Netherlands
关键词
HER2; exon20; poziotinib;
D O I
暂无
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
MA13.09
引用
收藏
页码:S147 / S148
页数:2
相关论文
共 50 条
  • [21] High activity of poziotinib in G778_P780dup HER2 exon 20 insertion mutations in non-small cell lung cancer (NSCLC)
    Le, X.
    Sun, S.
    Haura, E.
    Bertino, E.
    Baik, C.
    Mamdani, H.
    Leu, S.
    Thiagalingam, A.
    Kokhreidze, J.
    Lebel, F.
    Socinski, M. A.
    ANNALS OF ONCOLOGY, 2022, 33 (07) : S1084 - S1085
  • [22] A phase 2 study of poziotinib in patients with HER2-positive metastatic breast cancer (MBC) who have received prior HER2 regimens for MBC
    Lathrop, K.
    Lucas, J.
    Vacirca, J. L.
    Bhat, G.
    Choi, M. R.
    Naughton, M.
    CANCER RESEARCH, 2017, 77
  • [23] Safety, tolerability and preliminary efficacy of poziotinib with twice daily strategy in EGFR/HER2 Exon 20 mutant non-small cell lung cancer
    Sacher, A.
    Le, X.
    Cornelissen, R.
    Shum, E.
    Suga, J.
    Socinski, M.
    Molina, J. R.
    Haura, E.
    Clarke, J.
    Bhat, G.
    Lebel, F.
    Garassino, M. C.
    ANNALS OF ONCOLOGY, 2021, 32 : S15 - S15
  • [24] Poziotinib overcomes de novo resistance of HER2 exon 20 mutations in NSCLC and other cancers: Preclinical studies and initial clinical testing
    Robichaux, Jacqulyne P.
    Elamin, Yasir Y.
    Tan, Zhi
    Negrao, Marelo Vailati
    Routbort, Mark
    Roeck, Brent
    Li, Shuai
    Liu, Shengwu
    Chen, Ting
    Ahnert, Jordi Rodon
    Diao, Lixia
    Nilsson, Monique B.
    Zhang, Shuxing
    Yang, Zane
    Wang, Jing
    Meric-Bernstam, Funda
    Wong, Kwok-Kin
    Heymach, John V.
    CANCER RESEARCH, 2018, 78 (13)
  • [25] Metastatic Breast Cancer Patient With Activating HER2 Exon 20 Insertion Mutation With Response to Poziotinib: Case Report of Compassionate Drug Use
    Pandey, Apurva
    Brufsky, Adam M.
    CLINICAL BREAST CANCER, 2019, 19 (01) : E7 - E11
  • [26] Anti-angiogenic Therapy or Immunotherapy? A Multicenter Study of Patients with Advanced NSCLC with EGFR / HER2 exon 20 Insertion Mutations
    Chu, T.
    Li, J.
    Xie, M.
    Zhao, R.
    Qiang, H.
    Chang, Q.
    Qian, J.
    Lu, H.
    Shen, Y.
    Han, Y.
    Su, C.
    JOURNAL OF THORACIC ONCOLOGY, 2023, 18 (11) : S628 - S628
  • [27] Novel drugs targeting EGFR and HER2 exon 20 mutations in metastatic NSCLC
    Baraibar, Iosune
    Mezquita, Laura
    Gil-Bazo, Ignacio
    Planchard, David
    CRITICAL REVIEWS IN ONCOLOGY HEMATOLOGY, 2020, 148
  • [28] JIN-A04, highly effective tyrosine kinase inhibitor targeting HER2 exon 20 insertion mutations in NSCLC
    Yu, Mi Ra
    Yun, Mi Ran
    Lee, Jii Bum
    Lee, Ji Yun
    Aum, So Won
    Choi, Su Jin
    Park, Ju Yeon
    Oh, Seung Yeon
    Lee, Eun Ji
    Duggirala, Krishna Babu
    Lee, Kwangho
    Hong, Min Hee
    Lim, Sun Min
    Jo, Anna
    Seah, Ethan
    Kim, Choonok
    Cho, Byoung Chul
    CANCER RESEARCH, 2023, 83 (07)
  • [29] A phase 2 study of poziotinib in patients with EGFR or HER2 exon 20 mutation-positive non-small cell lung cancer
    Yang, Zandong
    Tchekmedyian, Nishan
    Chu, David T.
    Reddy, Guru
    Bhat, Gajanan
    Socinski, Mark A.
    JOURNAL OF CLINICAL ONCOLOGY, 2018, 36 (15)
  • [30] Efficacy and safety of sunvozertinib in treatment naive NSCLC patients with EGFR exon20 insertion mutations
    Xu, Yan
    Yang, James Chih-Hsin
    Chiu, Chao-Hua
    Hsu, Ping-Chih
    Mitchell, Paul
    Chang, Chia Lun
    John, Tom
    Bazhenova, Lyudmila
    Kim, Tae Min
    Yip, Ching Wan
    Wang, Mengzhao
    Janne, Pasi A.
    Zhou, Caicun
    JOURNAL OF CLINICAL ONCOLOGY, 2023, 41 (16)