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- [21] Development of a Commercial Manufacturing Process for Sotorasib, a First-in-Class KRASG12C InhibitorORGANIC PROCESS RESEARCH & DEVELOPMENT, 2022, 26 (11) : 3115 - 3125Zhang, Liang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAGriffin, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USABeaver, Matthew G.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USABlue, Laura E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USABorths, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USABrown, Derek B.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USACaille, Seb论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAChen, Ying论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USACherney, Alan H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USACochran, Brian M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAColyer, John T.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USACorbett, Michael T.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USACorrell, Tiffany L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USACrockett, Richard D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USADai, Xi-Jie论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USADornan, Peter K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAFarrell, Robert P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAHedley, Simon J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAHsieh, Hsiao-Wu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAHuang, Liang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAHuggins, Seth论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USALiu, Min论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USALovette, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAQuasdorf, Kyle论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAPowazinik, William论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAReifman, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USARobinson, Jo Anna论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USASangodkar, Rahul P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USASharma, Sonika论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAKumar, Srividya Sharvan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USASmith, Austin G.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USASt-Pierre, Gabrielle论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USATedrow, Jason S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Prepivotal Attribute Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAThiel, Oliver R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USATruong, Jonathan V.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAWalker, Shawn D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAWei, Carolyn S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAWilsily, Ashraf论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAXie, Yong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAYang, Ning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USAParsons, Andrew T.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA Amgen Inc, Pivotal & Commercial Synthet, Cambridge, MA 02142 USA
- [22] A Novel Inhibitor for KRASG12C Mutant Lung CarcinomaJOURNAL OF THORACIC ONCOLOGY, 2020, 15 (02) : S15 - S15Khan, H. Y.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USALi, Y.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USAAboukameel, A.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USAMpilla, G.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USASexton, R.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USAKanbur, T.论文数: 0 引用数: 0 h-index: 0机构: Izmir Inst Technol, Izmir, Turkey Wayne State Univ, Karmanos Canc Inst, Detroit, MI USACetinkaya, H.论文数: 0 引用数: 0 h-index: 0机构: Izmir Inst Technol, Izmir, Turkey Wayne State Univ, Karmanos Canc Inst, Detroit, MI USACagir, A.论文数: 0 引用数: 0 h-index: 0机构: Izmir Inst Technol, Izmir, Turkey Wayne State Univ, Karmanos Canc Inst, Detroit, MI USAAl-Hallak, M. N.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USASukari, A.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USAAzmi, A. S.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USANagasaka, M.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA Wayne State Univ, Karmanos Canc Inst, Detroit, MI USA
- [23] Gene expression correlates of adagrasib response in KRASG12C mutated non-small cell lung cancer (NSCLC)JOURNAL OF CLINICAL ONCOLOGY, 2024, 42 (16)Kim, Eejung论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USATong, Xinyuan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USAPatel, Ayushi论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USALiu, Shengwu论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USA论文数: 引用数: h-index:机构:Hover, Laura论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USAMukhopadhyay, Suman论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USASherman, Fiona论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USAChristensen, James G.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USAOlson, Peter论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USAAguirre, Andrew论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USAWong, Kwok论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USAJi, Hongbin论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA USA
- [24] Acquired Resistance to KRASG12C Inhibition in CancerNEW ENGLAND JOURNAL OF MEDICINE, 2021, 384 (25) : 2382 - 2393Awad, M. M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USALiu, S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Boston, MA 02115 USARybkin, I. I.论文数: 0 引用数: 0 h-index: 0机构: Henry Ford Canc Inst, Detroit, MI USA Dana Farber Canc Inst, Boston, MA 02115 USAArbour, K. C.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Dana Farber Canc Inst, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Zhu, V. W.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Sch Med, Chao Family Comprehens Canc Ctr, Orange, CA 92668 USA Dana Farber Canc Inst, Boston, MA 02115 USAJohnson, M. L.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Tennessee Oncol OneOncol, Nashville, TN USA Dana Farber Canc Inst, Boston, MA 02115 USAHeist, R. S.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Dana Farber Canc Inst, Boston, MA 02115 USAPatil, T.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Aurora, CO USA Dana Farber Canc Inst, Boston, MA 02115 USARiely, G. J.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Dana Farber Canc Inst, Boston, MA 02115 USAJacobson, J. O.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAYang, X.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Boston, MA 02115 USAPersky, N. S.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Boston, MA 02115 USARoot, D. E.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Boston, MA 02115 USALowder, K. E.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAFeng, H.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAZhang, S. S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Sch Med, Chao Family Comprehens Canc Ctr, Orange, CA 92668 USA Dana Farber Canc Inst, Boston, MA 02115 USAHaigis, K. M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Boston, MA 02115 USAHung, Y. P.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Dana Farber Canc Inst, Boston, MA 02115 USASholl, L. M.论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, 75 Francis St, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAWolpin, B. M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAWiese, J.论文数: 0 引用数: 0 h-index: 0机构: Boundless Bio, La Jolla, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAChristiansen, J.论文数: 0 引用数: 0 h-index: 0机构: Boundless Bio, La Jolla, CA USA Dana Farber Canc Inst, Boston, MA 02115 USALee, J.论文数: 0 引用数: 0 h-index: 0机构: Fdn Med, Cambridge, MA USA Dana Farber Canc Inst, Boston, MA 02115 USASchrock, A. B.论文数: 0 引用数: 0 h-index: 0机构: Fdn Med, Cambridge, MA USA Dana Farber Canc Inst, Boston, MA 02115 USALim, L. P.论文数: 0 引用数: 0 h-index: 0机构: Resolut Biosci, Kirkland, WA USA Dana Farber Canc Inst, Boston, MA 02115 USAGarg, K.论文数: 0 引用数: 0 h-index: 0机构: Resolut Biosci, Kirkland, WA USA Dana Farber Canc Inst, Boston, MA 02115 USALi, M.论文数: 0 引用数: 0 h-index: 0机构: Resolut Biosci, Kirkland, WA USA Dana Farber Canc Inst, Boston, MA 02115 USAEngstrom, L. D.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAWaters, L.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USALawson, J. D.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAOlson, P.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USALito, P.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Dana Farber Canc Inst, Boston, MA 02115 USAOu, S. -H. I.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Sch Med, Chao Family Comprehens Canc Ctr, Orange, CA 92668 USA Dana Farber Canc Inst, Boston, MA 02115 USAChristensen, J. G.论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAJanne, P. A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAAguirre, A. J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Brigham & Womens Hosp, 75 Francis St, Boston, MA 02115 USA Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Dana Farber Canc Inst, Boston, MA 02115 USA
- [25] Resistance to KRASG12C Inhibitors in Non-Small Cell Lung CancerFRONTIERS IN ONCOLOGY, 2021, 11Blaquier, Juan Bautista论文数: 0 引用数: 0 h-index: 0机构: Ctr Med Educ & Clin Res CEMIC, Thorac Oncol Unit, Med Oncol, Buenos Aires, DF, Argentina Ctr Med Educ & Clin Res CEMIC, Thorac Oncol Unit, Med Oncol, Buenos Aires, DF, ArgentinaCardona, Andres Felipe论文数: 0 引用数: 0 h-index: 0机构: Luis Carlos Sarmiento Angulo Canc Treatment & Res, Bogota, Colombia Fdn Clin & Appl Canc Res FICMAC, Bogota, Colombia Univ El Bosque, Mol Oncol & Biol Syst Res Grp FOX G ONCOLGrp, Bogota, Colombia Ctr Med Educ & Clin Res CEMIC, Thorac Oncol Unit, Med Oncol, Buenos Aires, DF, ArgentinaRecondo, Gonzalo论文数: 0 引用数: 0 h-index: 0机构: Ctr Med Educ & Clin Res CEMIC, Thorac Oncol Unit, Med Oncol, Buenos Aires, DF, Argentina Ctr Med Educ & Clin Res CEMIC, Thorac Oncol Unit, Med Oncol, Buenos Aires, DF, Argentina
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