共 58 条
NiFe-layered double hydroxide nanoparticle for co-delivery of DOX and siRNA to overcome multidrug resistance in MCF-7/ADR cells
被引:10
作者:

Bao, Yan-Ni
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机构:
Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China
Affiliated Hosp Shandong Med Coll, Pharm Dept, Linyi 276002, Shandong, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Xie, Xiu-Li
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h-index: 0
机构:
Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Lu, Li-Li
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Liu, Wen-Hao
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机构:
Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Ma, Yu-Chen
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Ke, Yi-Jun
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Ren, Huan
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Tan, Li-Na
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Wu, Li-Fang
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Song, Jue
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h-index: 0
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Jin, Yong
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h-index: 0
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Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China

Liu, Xiao-Yan
论文数: 0 引用数: 0
h-index: 0
机构:
Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
机构:
[1] Anhui Med Univ, Sch Pharm, Key Lab Antiinflammatory & Immune Med, Minist Educ, Hefei 230032, Peoples R China
[2] Inflammat & Immune Mediated Dis Lab Anhui Prov, Hefei 230032, Peoples R China
[3] Affiliated Hosp Shandong Med Coll, Pharm Dept, Linyi 276002, Shandong, Peoples R China
关键词:
Multidrug resistance (MDR);
Breast cancer resistance protein (BCRP);
Layered double hydroxide (LDH);
Doxorubicin (DOX);
siRNA;
BREAST-CANCER;
FACILE SYNTHESIS;
DRUG-RESISTANCE;
ANTICANCER DRUG;
CYCLE ARREST;
IN-SITU;
GENE;
DOXORUBICIN;
TUMOR;
EXPRESSION;
D O I:
10.1016/j.jddst.2023.104829
中图分类号:
R9 [药学];
学科分类号:
1007 ;
摘要:
Multidrug resistance (MDR) continues to be the major limiting factor in the cure of patients with cancer. Studies have shown that tumor multidrug resistance may be closely related to the multidrug-resistant protein secreted by itself, such as breast cancer resistance protein (BCRP). Therefore, inhibiting the production of multidrug-resistant proteins through genetic intervention may reverse tumor drug resistance. Herein, we use layered double hy-droxide nanoparticles (LDH) to co-deliver DOX and siRNA targeting BCRP RNA to reverse the resistance of MCF-7/ADR cells and enhance the anticancer activity of doxorubicin (DOX). In this platform, DOX is encapsulated in the nanoparticles, which have the characteristics of high drug loading and strong controlled-release, and siRNA is tightly adsorbed on the surface of the nanoparticles through electrostatic action to avoid the degradation of siRNA. Moreover, NiFe-LDH shows excellent ability to deliver siRNA and DOX into cells and enhance the internalization of siRNA and DOX. The experiment further confirms that siRNA-DOX@NiFe-LDH (1:1) shows an effective gene silencing effect and down-regulated the expression of BCRP. In vitro experiments show that siRNA-DOX@NiFe-LDH inhibits cell proliferation by affecting the cell cycle and inducing apoptosis. In vivo experi-ments, MCF-7/ADR xenotransplantation therapy also reveals that siRNA-DOX@NiFe-LDH has a significant antitumor effect. We believe that this work has great potential for reversing the drug resistance of breast cancer and improving the effectiveness of chemotherapy.
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页数:10
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Kilchrist, Kameron V.
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PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
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Sarett, Samantha M.
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Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA

Werfel, Thomas A.
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Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA

Lee, Linus
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Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA

Jackson, Meredith A.
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Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA

Kilchrist, Kameron V.
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Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA

Brantley-Sieders, Dana
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Vanderbilt Univ, Med Ctr, Dept Med, Nashville, TN 37232 USA Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA

Duvall, Craig L.
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Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA Vanderbilt Univ, Dept Biomed Engn, Nashville, TN 37235 USA
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Modulation of Intestinal Transport and Absorption of Topotecan, a BCRP Substrate, by Various Pharmaceutical Excipients and Their Inhibitory Mechanisms of BCRP Transporter
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Sakane, Toshiyasu
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JOURNAL OF PHARMACEUTICAL SCIENCES,
2019, 108 (03)
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Sawangrat, Kasirawat
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机构:
Kyoto Pharmaceut Univ, Dept Biopharmaceut, Yamashina Ku, Misasagi, Kyoto 6078414, Japan Kyoto Pharmaceut Univ, Dept Biopharmaceut, Yamashina Ku, Misasagi, Kyoto 6078414, Japan

Yamashita, Shugo
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Kobe Pharmaceut Univ, Dept Pharmaceut Technol, Higashinada Ku, Kobe, Hyogo 6588558, Japan Kyoto Pharmaceut Univ, Dept Biopharmaceut, Yamashina Ku, Misasagi, Kyoto 6078414, Japan

Tanaka, Akiko
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Kobe Pharmaceut Univ, Dept Pharmaceut Technol, Higashinada Ku, Kobe, Hyogo 6588558, Japan Kyoto Pharmaceut Univ, Dept Biopharmaceut, Yamashina Ku, Misasagi, Kyoto 6078414, Japan

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Katsumi, Hidemasa
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Kyoto Pharmaceut Univ, Dept Biopharmaceut, Yamashina Ku, Misasagi, Kyoto 6078414, Japan Kyoto Pharmaceut Univ, Dept Biopharmaceut, Yamashina Ku, Misasagi, Kyoto 6078414, Japan

Sakane, Toshiyasu
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Kobe Pharmaceut Univ, Dept Pharmaceut Technol, Higashinada Ku, Kobe, Hyogo 6588558, Japan Kyoto Pharmaceut Univ, Dept Biopharmaceut, Yamashina Ku, Misasagi, Kyoto 6078414, Japan

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