共 25 条
- [1] 1-(4-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)-3-methoxyphenyl)-3-(2-(dimethylamino)ethyl)imidazolidin-2-one (ZX-42), a novel ALK inhibitor, induces apoptosis and protective autophagy in H2228 cellsJOURNAL OF PHARMACY AND PHARMACOLOGY, 2020, 72 (10) : 1370 - 1382Wang, Lijing论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaXu, Xiaobo论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaLiu, Tong论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaWang, Junfang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaShen, Jiwei论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaGuo, Ming论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaWu, Yingliang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaZhai, Xin论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaZuo, Daiying论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China
- [2] 1-(4-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl) amino)-3-methoxyphenyl)-3-(2-(dimethylamino)ethyl)imidazolidin-2-one (ZX-42) inhibits cell proliferation and induces apoptosis via inhibiting ALK and its downstream pathways in Karpas299 cellsTOXICOLOGY AND APPLIED PHARMACOLOGY, 2022, 450Chang, Xing论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaWang, Junfang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaBian, Jiang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaLiu, Zi论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaGuo, Ming论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaLi, Zengqiang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaWu, Yingliang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaZhai, Xin论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaZuo, Daiying论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China
- [3] Discovery of a potent EGFR and ALK dual mutation inhibitor containing N-(3-((4-((2-(cyclopropylsulfinyl)phenyl)amino)pyrimidin-2-yl)amino) phenyl)acrylamide scaffoldBIOORGANIC CHEMISTRY, 2022, 129Li, Wei论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaYao, Han论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaGu, Chenxi论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaRen, Yuanyuan论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaLiu, Jiadai论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaAn, Baijiao论文数: 0 引用数: 0 h-index: 0机构: Binzhou Med Univ, Sch Pharmaceut Sci, Yantai 264003, Shandong, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaHu, Wenhao论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaLi, Xingshu论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R ChinaChan, Albert S. C.论文数: 0 引用数: 0 h-index: 0机构: Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China Sun Yat Sen Univ, Sch Pharmaceut Sci, Guangzhou 510006, Peoples R China
- [4] Discovery of N-(5-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)-4-methoxy-2-(4-methyl-1,4-diazepan-1-yl)phenyl)acrylamide (CHMFL-ALK/EGFR-050) as a potent ALK/EGFR dual kinase inhibitor capable of overcoming a variety of ALK/EGFR associated drug resistant mutants in NSCLCEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 139 : 674 - 697Chen, Yongfei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWu, Jiaxin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230026, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Aoli论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaQi, Ziping论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaJiang, Taoshan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Anhui Agr Univ, Sch Life Sci, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaChen, Cheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230026, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaZou, Fengming论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaHu, Chen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230026, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Wei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWu, Hong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaHu, Zhenquan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Wenchao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Beilei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230026, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Li论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230026, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaRen, Tao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Hefei Inst Phys Sci, Inst Technol Innovat, Precis Targeted Therapy Discovery Ctr, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaZhang, Shanchun论文数: 0 引用数: 0 h-index: 0机构: CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Hefei Cosource Med Technol Co LTD, 358 Ganquan Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Qingsong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230026, Anhui, Peoples R China Chinese Acad Sci, Hefei Inst Phys Sci, Inst Technol Innovat, Precis Targeted Therapy Discovery Ctr, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Jing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China
- [5] 5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-((4-methylpiperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)phenyl)pyrimidine-2,4-diamine (WY-135), a novel ALK inhibitor, induces cell cycle arrest and apoptosis through inhibiting ALK and its downstream pathways in Karpas299 and H2228 cellsCHEMICO-BIOLOGICAL INTERACTIONS, 2018, 284 : 24 - 31Han, Mengting论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaShen, Jiwei论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaWang, Lijing论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaWang, Yu论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaZhai, Xin论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaLi, Yao论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaLiu, Meiqiao论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaLi, Zengqiang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaZuo, Daiying论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaWu, Yingliang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China
- [6] 5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-((4-methylpiperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)phenyl)pyrimidine-2,4-diamine (WY-135), a novel ALK inhibitor, induces cell cycle arrest and apoptosis through inhibiting ALK and its downstream pathways in Karpas299 and H2228 cells (vol 284, pg 24, 2018)CHEMICO-BIOLOGICAL INTERACTIONS, 2022, 356Han, Mengting论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaShen, Jiwei论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaWang, Lijing论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaWang, Yu论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaZhai, Xin论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaLi, Yao论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaLiu, Meiqiao论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaGao, Meiqi论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaLi, Zengqiang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaZuo, Daiying论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R ChinaWu, Yingliang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Dept Pharmacol, 103 Wenhua Rd, Shenyang 110016, Peoples R China
- [7] Discovery of 4-(4-(3-(1-(2-(piperidin-1-yl)ethyl)-1H-benzo[d] imidazole-2-yl)isoxazol-5-yl)phenyl)morpholine as a novel c-Myc inhibitor against lung cancer in vitro and in vivoEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 281Gao, Jian论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaYin, Jiacheng论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaLi, Shihao论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaJia, Pingting论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaHong, Renjie论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaChen, Jiahui论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaQu, Xinxin论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaZhang, Zihui论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaLi, Mengting论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R ChinaZhao, Hui论文数: 0 引用数: 0 h-index: 0机构: Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China Anhui Univ Sci & Technol, Sch Med, Huainan, Peoples R China
- [8] SYNTHESIS, CHARACTERIZATION AND ANTIMICROBIAL EVALUATION OF NOVEL COMPOUNDS OF 3-((BENZO[D]THIAZOL-2-YLMETHYL)AMINO)-1-(2,5- DIFLUOROBENZOYL)-4-(2-(4-(SUBSTITUTED )PHENYL)HYDRAZONO)-1H- PYRAZOL-5(4H)-ONEHETEROCYCLIC LETTERS, 2018, 8 (04): : 805 - 813Kumari, M. Swarna论文数: 0 引用数: 0 h-index: 0机构: Sri Krishnadevaraya Univ, Dept Chem, Anantapur, Andhra Pradesh, India Sri Krishnadevaraya Univ, Dept Chem, Anantapur, Andhra Pradesh, IndiaRavindhranath, L. K.论文数: 0 引用数: 0 h-index: 0机构: Sri Krishnadevaraya Univ, Dept Chem, Anantapur, Andhra Pradesh, IndiaBabu, K. Sudhakar论文数: 0 引用数: 0 h-index: 0机构: Sri Krishnadevaraya Univ, Dept Chem, Anantapur, Andhra Pradesh, IndiaReddy, K. Ashok vardhan论文数: 0 引用数: 0 h-index: 0机构: Dr KV Subba Reddy Coll Engn Women, Kurnool, AP, India Sri Krishnadevaraya Univ, Dept Chem, Anantapur, Andhra Pradesh, India
- [9] Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibitor for PDGFRα driving chronic eosinophilic leukemiaEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 150 : 366 - 384Wang, Qiang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Feiyang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaQi, Shuang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaQi, Ziping论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaYan, Xiao-E.论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Hlth Sci Ctr, Sch Basic Med Sci, Inst Syst Biomed,Dept Biophys, Beijing 100191, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Beilei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Aoli论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Wei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaChen, Cheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Xiaochuan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaJiang, Zongru论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaHu, Zhenquan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Li论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Wenchao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaRen, Tao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Hefei Inst Phys Sci, Inst Technol Innovat, Precis Targeted Therapy Discovery Ctr, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaZhang, Shanchun论文数: 0 引用数: 0 h-index: 0机构: CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Hefei Cosource Med Technol Co LTD, 358 Ganquan Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaYun, Cai-Hong论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Hlth Sci Ctr, Sch Basic Med Sci, Inst Syst Biomed,Dept Biophys, Beijing 100191, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Qingsong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, Hefei Sci Ctr, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Jing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China CHMFL HCMTC Target Therapy Joint Lab, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, Hefei Sci Ctr, 350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Chinese Acad Sci, High Magnet Field Lab, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China
- [10] Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino) pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignanciesEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 173 : 44 - 62Tong, Lexian论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaSong, Pinrao论文数: 0 引用数: 0 h-index: 0机构: Shanghai Haini Pharmaceut Co Ltd, Yangtze River Pharmaceut Grp, Shanghai 201318, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaJiang, Kailong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Natl Ctr Drug Screening, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaXu, Lei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Natl Ctr Drug Screening, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China ShanghaiTech Univ, Shanghai 201210, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaJin, Tingting论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, 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310058, Zhejiang, Peoples R ChinaGao, Anhui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Natl Ctr Drug Screening, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaZhou, Yubo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Natl Ctr Drug Screening, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaLiu, Tao论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaLi, Jia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Natl Ctr Drug Screening, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China ShanghaiTech Univ, Shanghai 201210, Peoples R China Pilot Natl Lab Marine Sci & Technol Qingdao, Open Studio Druggabil Res Marine Nat Prod, 1 Wenhai Rd, Qingdao 266237, Shandong, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R ChinaHu, Yongzhou论文数: 0 引用数: 0 h-index: 0机构: Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China Zhejiang Univ, Coll Pharmaceut Sci, Zhejiang Prov Key Lab Anticanc Drug Res, ZJU ENS Joint Lab Med Chem, Hangzhou 310058, Zhejiang, Peoples R China