共 36 条
[31]
Antibacterial and antibiotic modifying activity of chalcone (2E)-1-(4'-aminophenyl)-3-(4-methoxyphenyl)-prop-2-en-1-one in strains of Staphylococcus aureus carrying NorA and MepA efflux pumps: In vitro and in silico approaches
[J].
Silva, Jacilene
;
Rocha, Janaina Esmeraldo
;
Xavier, Jayze da Cunha
;
de Freitas, Thiago Sampaio
;
Coutinho, Henrique Douglas Melo
;
Bandeira, Paulo Nogueira
;
de Oliveira, Mateus Rodrigues
;
da Rocha, Matheus Nunes
;
Marinho, Emanuelle Machado
;
Monteiro, Norberto de Kassio Vieira
;
Ribeiro, Lyanna Rodrigues
;
de Menezes, Ramon Roseo Paula Pessoa Bezerra
;
Marinho, Marcia Machado
;
Teixeira, Alexandre Magno Rodrigues
;
dos Santos, Helcio Silva
;
Marinho, Emmanuel Silva
.
MICROBIAL PATHOGENESIS,
2022, 169

Silva, Jacilene
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Rocha, Janaina Esmeraldo
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机构:
Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Xavier, Jayze da Cunha
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Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

de Freitas, Thiago Sampaio
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机构:
Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Coutinho, Henrique Douglas Melo
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机构:
Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Bandeira, Paulo Nogueira
论文数: 0 引用数: 0
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机构:
Univ Estadual Vale Acarau, Ctr Ciencias Exatas & Tecnol, Sobral, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

de Oliveira, Mateus Rodrigues
论文数: 0 引用数: 0
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机构:
Univ Estadual Vale Acarau, Ctr Ciencias Exatas & Tecnol, Sobral, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

da Rocha, Matheus Nunes
论文数: 0 引用数: 0
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机构:
Univ Estadual Ceara, Fac Filosofia Dom Aureliano Matos, Limoeiro Norte, Limoeiro Do Norte, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Marinho, Emanuelle Machado
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h-index: 0
机构:
Univ Fed Ceara, Dept Quim Analit & Fis Quim, Fortaleza, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Monteiro, Norberto de Kassio Vieira
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机构:
Univ Fed Ceara, Dept Quim Analit & Fis Quim, Fortaleza, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Ribeiro, Lyanna Rodrigues
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Fed Ceara, Dept Anal Clin & Toxicol, Fortaleza, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

de Menezes, Ramon Roseo Paula Pessoa Bezerra
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Fed Ceara, Dept Anal Clin & Toxicol, Fortaleza, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Marinho, Marcia Machado
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Estadual Vale Acarau, Ctr Ciencias Exatas & Tecnol, Sobral, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Teixeira, Alexandre Magno Rodrigues
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

dos Santos, Helcio Silva
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil
Univ Estadual Vale Acarau, Ctr Ciencias Exatas & Tecnol, Sobral, CE, Brazil
Univ Estadual Ceara, Ctr Ciencias & Tecnol, Programa Posgrad Ciencias Nat, Fortaleza, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil

Marinho, Emmanuel Silva
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Estadual Ceara, Fac Filosofia Dom Aureliano Matos, Limoeiro Norte, Limoeiro Do Norte, CE, Brazil
Univ Estadual Ceara, Ctr Ciencias & Tecnol, Programa Posgrad Ciencias Nat, Fortaleza, CE, Brazil
Univ Estadual Ceara Limoeiro Norte, 850 Univ Ave, BR-62040370 Sobral, CE, Brazil Univ Reg Cariri, Dept Quim Biol, Crato, CE, Brazil
[32]
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search
[J].
Cedraro, Nicholas
;
Cannalire, Rolando
;
Astolfi, Andrea
;
Mangiaterra, Gianmarco
;
Felicetti, Tommaso
;
Vaiasicca, Salvatore
;
Cernicchi, Giada
;
Massari, Serena
;
Manfroni, Giuseppe
;
Tabarrini, Oriana
;
Cecchetti, Violetta
;
Barreca, Maria Letizia
;
Biavasco, Francesca
;
Sabatini, Stefano
.
CHEMMEDCHEM,
2021, 16 (19)
:3044-3059

Cedraro, Nicholas
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Cannalire, Rolando
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Napoli Federico II, Dept Pharm, Via D Montesano 49, I-80131 Naples, Italy
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Astolfi, Andrea
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h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Mangiaterra, Gianmarco
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Felicetti, Tommaso
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Vaiasicca, Salvatore
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

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Massari, Serena
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Manfroni, Giuseppe
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Tabarrini, Oriana
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Cecchetti, Violetta
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Barreca, Maria Letizia
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Biavasco, Francesca
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy

Sabatini, Stefano
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dept Pharmaceut Sci, Via Liceo 1, I-06123 Perugia, Italy Univ Politecn Marche, Dept Life & Environm Sci, Via Brecce Bianche, I-60131 Ancona, Italy
[33]
Synthesis of Some Novel 4-bromobenzoic Acid Clubbed Hydrazone Schiff Base Derivatives as Potent α-amylase Inhibitors: In vitro and In silico Studies
[J].
Khan, Momin
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Alam, Faima
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Alam, Aftab
;
Wadood, Abdul
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Shams, Sulaiman
;
Ali, Mahboob
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Shah, Sana
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Alasmari, Abdullah F.
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Alharbi, Metab
;
Alasmari, Fawaz
.
LETTERS IN DRUG DESIGN & DISCOVERY,
2024, 21 (15)
:3186-3197

Khan, Momin
论文数: 0 引用数: 0
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机构:
Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

Alam, Faima
论文数: 0 引用数: 0
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机构:
Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

Alam, Aftab
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Malakand, Dept Chem, Chakdara 18800, Lower Dir, Pakistan Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

Wadood, Abdul
论文数: 0 引用数: 0
h-index: 0
机构:
Abdul Wali Khan Univ, Dept Biochem, Mardan 23200, Pakistan Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

论文数: 引用数:
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Ali, Mahboob
论文数: 0 引用数: 0
h-index: 0
机构:
Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

Shah, Sana
论文数: 0 引用数: 0
h-index: 0
机构:
Heilongjiang Univ, Sch Chem & Mat, Key Lab Funct Inorgan Mat Chem, Minist Educ, Harbin 150080, Peoples R China Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

Alasmari, Abdullah F.
论文数: 0 引用数: 0
h-index: 0
机构:
King Saud Univ, Coll Pharm, Dept Pharmacol & Toxicol, Riyadh 11451, Saudi Arabia Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

Alharbi, Metab
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h-index: 0
机构:
King Saud Univ, Coll Pharm, Dept Pharmacol & Toxicol, Riyadh 11451, Saudi Arabia Abdul Wali Khan Univ, Dept Chem, Mardan 23200, Pakistan

论文数: 引用数:
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[34]
Biofunctionalization of Poly(lactide-co-glycolic acid) Using Potent NorA Efflux Pump Inhibitors Immobilized on Nanometric Alpha-Zirconium Phosphate to Reduce Biofilm Formation
[J].
Pica, Monica
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Messere, Nicla
;
Felicetti, Tommaso
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Sabatini, Stefano
;
Pietrella, Donatella
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Nocchetti, Morena
.
MATERIALS,
2021, 14 (03)
:1-14

论文数: 引用数:
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Messere, Nicla
论文数: 0 引用数: 0
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机构:
Univ Perugia, Dipartimento Sci Farmaceut, Via Liceo 1, I-06123 Perugia, Italy Univ Perugia, Dipartimento Sci Farmaceut, Via Liceo 1, I-06123 Perugia, Italy

Felicetti, Tommaso
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机构:
Univ Perugia, Dipartimento Sci Farmaceut, Via Liceo 1, I-06123 Perugia, Italy Univ Perugia, Dipartimento Sci Farmaceut, Via Liceo 1, I-06123 Perugia, Italy

Sabatini, Stefano
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机构:
Univ Perugia, Dipartimento Sci Farmaceut, Via Liceo 1, I-06123 Perugia, Italy Univ Perugia, Dipartimento Sci Farmaceut, Via Liceo 1, I-06123 Perugia, Italy

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[35]
Evolution from a Natural Flavones Nucleus to Obtain 2-(4-Propoxyphenyl)quinoline Derivatives As Potent Inhibitors of the S. aureus NorA Efflux Pump
[J].
Sabatini, Stefano
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Gosetto, Francesca
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Manfroni, Giuseppe
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Tabarrini, Oriana
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Kaatz, Glenn W.
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Patel, Diixa
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Cecchetti, Violetta
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JOURNAL OF MEDICINAL CHEMISTRY,
2011, 54 (16)
:5722-5736

Sabatini, Stefano
论文数: 0 引用数: 0
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机构:
Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy

Gosetto, Francesca
论文数: 0 引用数: 0
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机构:
Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy

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Tabarrini, Oriana
论文数: 0 引用数: 0
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机构:
Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy

Kaatz, Glenn W.
论文数: 0 引用数: 0
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机构:
Wayne State Univ, Sch Med, Div Infect Dis, Dept Internal Med, Detroit, MI 48201 USA
John D Dingell Dept Vet Affairs Med Ctr, Detroit, MI 48201 USA Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy

Patel, Diixa
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h-index: 0
机构:
Wayne State Univ, Sch Med, Div Infect Dis, Dept Internal Med, Detroit, MI 48201 USA
John D Dingell Dept Vet Affairs Med Ctr, Detroit, MI 48201 USA Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy

Cecchetti, Violetta
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy Univ Perugia, Dipartimento Chim & Tecnol Farmaco, I-06123 Perugia, Italy
[36]
Discovery of 4-[(5-arylidene-4-oxothiazolidin-3-yl)methyl]benzoic acid derivatives active as novel potent allosteric inhibitors of protein tyrosine phosphatase 1B: In silico studies and in vitro evaluation as insulinomimetic and anti-inflammatory agents
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Ottana, Rosaria
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Paoli, Paolo
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Nass, Alexandra
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Lori, Giulia
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Cardile, Venera
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Adornato, Ilenia
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Rotondo, Archimede
;
Graziano, Adriana Carol Eleonora
;
Wolber, Gerhard
;
Maccari, Rosanna
.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,
2017, 127
:840-858

Ottana, Rosaria
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy

Paoli, Paolo
论文数: 0 引用数: 0
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机构:
Univ Florence, Dept Sci Biomed Sperimentali & Clin, Sez Sci Biochim, Viale Morgagni 50, I-50134 Florence, Italy Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy

Nass, Alexandra
论文数: 0 引用数: 0
h-index: 0
机构:
Free Univ Berlin, Inst Pharm, Comp Aided Mol Design, Koenigin Luisestr 2 4, D-14195 Berlin, Germany Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy

Lori, Giulia
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Florence, Dept Sci Biomed Sperimentali & Clin, Sez Sci Biochim, Viale Morgagni 50, I-50134 Florence, Italy Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy

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Adornato, Ilenia
论文数: 0 引用数: 0
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机构:
Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy

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Graziano, Adriana Carol Eleonora
论文数: 0 引用数: 0
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机构:
Univ Catania, Physiol Sect, Dept Biomed & Biotechnol Sci, Via S Sofia 64, I-95125 Catania, Italy Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy

Wolber, Gerhard
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h-index: 0
机构:
Free Univ Berlin, Inst Pharm, Comp Aided Mol Design, Koenigin Luisestr 2 4, D-14195 Berlin, Germany Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy

Maccari, Rosanna
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy Univ Messina, Polo Univ Annunziata, Dept Sci Chim Biol Farmaceut & Ambientali, Viale SS Annunziata, I-98168 Messina, Italy