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- [1] Novel, brain penetrant small molecule inhibitor of PD-L1 for targeting glioblastoma and brain metastasisEUROPEAN JOURNAL OF CANCER, 2022, 174 : S125 - S125Dhanalakshmi, S.论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USA Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USARajagopal, S.论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Discovery Chem, Bedminster, NJ USA Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USAGajendran, C.论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USA Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USASadhu, M. N.论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Discovery Chem, Bedminster, NJ USA Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USAZainuddin, M.论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USA Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USAGosu, R.论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Prot Chem, Bedminster, NJ USA Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USARastelli, L.论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USA Jubilant Therapeut Inc, Discovery Biol, Bedminster, NJ USA
- [2] NOVEL, BRAIN PENETRANT SMALL MOLECULE INHIBITOR OF PD-L1 FOR TARGETING GLIOBLASTOMA AND BRAIN METASTASISJOURNAL FOR IMMUNOTHERAPY OF CANCER, 2022, 10 : A1430 - A1430Sivanandhan, Dhanalakshmi论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USARajagopal, Sridharan论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USARajagopal, Sridharan论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USAGajendran, Chandru论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USASadhu, M. Naveen论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USAZainuddin, Mohammed论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USAGosu, Ramachandraiah论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USARastelli, Luca论文数: 0 引用数: 0 h-index: 0机构: Jubilant Therapeut Inc, Bedminster, NJ USA Jubilant Therapeut Inc, Bedminster, NJ USA
- [3] Discovery and characterization of a novel small molecule antagonist of PD-L1MOLECULAR CANCER THERAPEUTICS, 2019, 18 (12)Ying, Haiyan论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaYang, Fei论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaZhang, Mingming论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaZhang, Yongxian论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaZhao, Yuan论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaZhang, Lei论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaYu, Hongping论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaChen, Zhui论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R ChinaXu, Yao-chang论文数: 0 引用数: 0 h-index: 0机构: Abbisko Therapeut, Shanghai, Peoples R China Abbisko Therapeut, Shanghai, Peoples R China
- [4] Characterization of INCB086550: A Potent and Novel Small-Molecule PD-L1 InhibitorCANCER DISCOVERY, 2022, 12 (06) : 1482 - 1499Koblish, Holly K.论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAWu, Liangxing论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAWang, Liang-Chuan S.论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USALiu, Phillip C. C.论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAWynn, Richard论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USARios-Doria, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USASpitz, Susan论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USALiu, Hao论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAVolgina, Alla论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAZolotarjova, Nina论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAKapilashrami, Kanishk论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USABehshad, Elham论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USACovington, Maryanne论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAYang, Yan-Ou论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USALi, Jingwei论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USADiamond, Sharon论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USASoloviev, Maxim论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAO'Hayer, Kevin论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USARubin, Stephen论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAKanellopoulou, Chrysi论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAYang, Gengjie论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USARupar, Mark论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USADiMatteo, Darlise论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USALin, Luping论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAStevens, Christina论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAZhang, Yue论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAThekkat, Pramod论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAGeschwindt, Ryan论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAMarando, Cindy论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAYeleswaram, Swamy论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAJackson, Jeff论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAScherle, Peggy论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAHuber, Reid论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAYao, Wenqing论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USAHollis, Gregory论文数: 0 引用数: 0 h-index: 0机构: Incyte Res Inst, Wilmington, DE USA Incyte Res Inst, Wilmington, DE USA
- [5] Novel Small-Molecule PD-L1 Inhibitor Induces PD-L1 Internalization and Optimizes the Immune MicroenvironmentJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (03) : 2064 - 2083Sun, Chengliang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaYin, Mingxiao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci & Peking Union Med Coll, Inst Med Biotechnol, Beijing 100050, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaCheng, Yao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaKuang, Zean论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci & Peking Union Med Coll, Inst Med Biotechnol, Beijing 100050, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaLiu, Xiaojia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci & Peking Union Med Coll, Inst Med Biotechnol, Beijing 100050, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaWang, Gefei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaWang, Xiao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaYuan, Kai论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaMin, Wenjian论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaDong, Jingwen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci & Peking Union Med Coll, Inst Med Biotechnol, Beijing 100050, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaHou, Yi论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaHu, Lingrong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaZhang, Guoyu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaPei, Wenli论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaWang, Liping论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaSun, Yanze论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaYu, Xinmiao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaXiao, Yibei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaDeng, Hongbin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci & Peking Union Med Coll, Inst Med Biotechnol, Beijing 100050, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R ChinaYang, Peng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Jiangsu Key Lab Drug Design & Optimizat, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Pharmacol, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, Nanjing 210009, Peoples R China
- [6] In vitro characterization of a small molecule PD-1 inhibitor that targets the PD-l/PD-L1 interactionSCIENTIFIC REPORTS, 2022, 12 (01)论文数: 引用数: h-index:机构:Chung, Wei-Min论文数: 0 引用数: 0 h-index: 0机构: China Med Univ, Grad Inst Biomed Sci, Taichung 40403, Taiwan China Med Univ, PhD Program Biotechnol & Biomed Ind, Taichung 40403, Taiwan论文数: 引用数: h-index:机构:Cheng, Ju-Chien论文数: 0 引用数: 0 h-index: 0机构: China Med Univ, Dept Med Lab Sci & Biotechnol, Taichung 40403, Taiwan China Med Univ, PhD Program Biotechnol & Biomed Ind, Taichung 40403, TaiwanHsu, Kai-Cheng论文数: 0 引用数: 0 h-index: 0机构: Taipei Med Univ, Grad Inst Canc Biol & Drug Discovery, Taipei 11031, Taiwan Taipei Med Univ, PhD Program Canc Mol Biol & Drug Discovery, Taipei 11031, Taiwan China Med Univ, PhD Program Biotechnol & Biomed Ind, Taichung 40403, TaiwanTzeng, Huey-En论文数: 0 引用数: 0 h-index: 0机构: Taipei Med Univ, Grad Inst Canc Biol & Drug Discovery, Taipei 11031, Taiwan Taipei Med Univ, PhD Program Canc Mol Biol & Drug Discovery, Taipei 11031, Taiwan Taipei Med Univ Hosp, Dept Med, Div Hematol Oncol, Taipei 11031, Taiwan Taipei Med Univ, Sch Med, Taipei 11031, Taiwan Taichung Vet Gen Hosp, Dept Med Res, Taichung 40705, Taiwan Taichung Vet Gen Hosp, Div Hematol & Oncol, Taichung 40705, Taiwan China Med Univ, PhD Program Biotechnol & Biomed Ind, Taichung 40403, Taiwan
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