共 169 条
Therapeutic resistance to anti-oestrogen therapy in breast cancer
被引:91
作者:

Will, Marie
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA
Mem Sloan Kettering Canc Ctr, Dept Med, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA

Liang, Jackson
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Oncol Biomarker Dev, South San Francisco, CA USA Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA

Metcalfe, Ciara
论文数: 0 引用数: 0
h-index: 0
机构:
Genentech Inc, Dept Discovery Oncol, South San Francisco, CA 94080 USA Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA

Chandarlapaty, Sarat
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA
Mem Sloan Kettering Canc Ctr, Dept Med, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA
机构:
[1] Mem Sloan Kettering Canc Ctr, Human Oncol & Pathogenesis Program, New York, NY 10065 USA
[2] Mem Sloan Kettering Canc Ctr, Dept Med, New York, NY 10065 USA
[3] Genentech Inc, Dept Oncol Biomarker Dev, South San Francisco, CA USA
[4] Genentech Inc, Dept Discovery Oncol, South San Francisco, CA 94080 USA
基金:
美国国家卫生研究院;
关键词:
ESTROGEN-RECEPTOR-ALPHA;
CELL-CYCLE PROGRESSION;
ACQUIRED ENDOCRINE RESISTANCE;
ACTIVATING ESR1 MUTATIONS;
GROWTH-FACTOR;
AROMATASE INHIBITORS;
POSTMENOPAUSAL WOMEN;
CDK4/6;
INHIBITORS;
ELACESTRANT RAD1901;
ANTITUMOR-ACTIVITY;
D O I:
10.1038/s41568-023-00604-3
中图分类号:
R73 [肿瘤学];
学科分类号:
100214 ;
摘要:
Although selective antagonism of oestrogen receptor signalling in breast cancer has been one of the most successful therapeutic approaches in oncology, resistance is a major clinical challenge. In this Review, Will et al. explore mechanisms of oestrogen-receptor-& alpha;-targeted therapeutic resistance and strategies to overcome it. The hormone receptor oestrogen receptor-& alpha; (ER) orchestrates physiological mammary gland development, breast carcinogenesis and the progression of breast tumours into lethal, treatment-refractory systemic disease. Selective antagonism of ER signalling has been one of the most successful therapeutic approaches in oncology, benefiting patients as both a cancer preventative measure and a cancer treatment strategy. However, resistance to anti-oestrogen therapy is a major clinical challenge. Over the past decade, we have gained an understanding of how breast cancers evolve under the pressure of anti-oestrogen therapy. This is best depicted by the case of oestrogen-independent mutations in the gene encoding ER (ESR1), which are virtually absent in primary breast cancer but highly prevalent (20-40%) in anti-oestrogen-treated metastatic disease. These and other findings highlight the 'evolvability' of ER+ breast cancer and the need to understand molecular processes by which this evolution occurs. Recent development and approval of next-generation ER antagonists to target ESR1-mutant breast cancer underscores the clinical importance of this evolvability and sets a new paradigm for the treatment of ER+ breast cancers.
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页码:673 / 685
页数:13
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Yu, Jiajie
;
Metcalfe, Ciara
;
De Bruyn, Tom
;
Gelzleichter, Thomas
;
Malhi, Vikram
;
Perez-Moreno, Pablo D.
;
Wang, Xiaojing
.
EXPERT OPINION ON INVESTIGATIONAL DRUGS,
2022, 31 (06)
:515-529

Chen, Ya-Chi
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机构:
Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA

Yu, Jiajie
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Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA

Metcalfe, Ciara
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Genentech Inc, Discovery Oncol, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA

De Bruyn, Tom
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h-index: 0
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Genentech Inc, Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA

Gelzleichter, Thomas
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Genentech Inc, Genentech Res & Early Dev, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA

Malhi, Vikram
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Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA

Perez-Moreno, Pablo D.
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Genentech Inc, Prod Dev Oncol, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA

Wang, Xiaojing
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h-index: 0
机构:
Genentech Inc, Discovery Chem, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, Clin Pharmacol, 1 DNA Way, San Francisco, CA 94080 USA