Design, synthesis and insecticidal activity of biphenyl-diamide derivatives

被引:1
|
作者
Ye Liu [1 ]
Chao Lei [1 ]
Xiao-Yong Xu [1 ]
Xu-Sheng Shao [1 ]
Zhong Li [1 ]
机构
[1] Shanghai Key Laboratory of Chemical Biology,School of Pharmacy,East China University of Science and Technology
关键词
Diamide; Insecticide; Ryanodine insecticide; Biphenyl;
D O I
暂无
中图分类号
TQ453 [杀虫剂];
学科分类号
090403 ;
摘要
Diamides acting on insect ryanodine receptors are an intensive research area now. In order to search for novel candidates, a series of diamides containing biphenyl substructure were designed and synthesized.Their insecticidal activities against armyworms(Mythimna sepatara) and aphis(Aphis craccivora) were screened. The compounds with 3,5-dichloro-4-(1,1,2,2-tetrafluoroethoxy)phenyl substituent were found to be insecticidal to armyworms with the similar symptoms to poisoning by flubendiamide. In this research, we presented a novel type of diamide insecticide as a lead compound for further optimization.
引用
收藏
页码:321 / 324
页数:4
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