A convenient one-pot three component synthesis of 3-aminoalkylated indoles catalyzed by 3-chlorophenylboronic acid

被引：0

作者：

Santosh V.Goswami

Prashant.B.Thorat

Vijay N.Kadam

Sachin A.Khiste

Sudhakar R.Bhusare

机构：

[1] DepartmentofChemistry,DnyanopasakCollege

来源：

Chinese Chemical Letters | 2013年 / 24卷 / 05期

关键词：

3-Aminoalkylaed indoles; 3-Chlorophenylboronic acid; Aromatic aldehyde; N-Methylaniline; Indoles;

D O I：

暂无

中图分类号：

O643.32 [催化反应];

学科分类号：

081705 ;

摘要：

<正>An efficient protocol was developed for the synthesis of 3-aminoalkylated indoles using 3- chlorophenylboronic acid as a catalyst under ambient temperature conditions.The three-component reaction of indoles,aromatic aldehydes and N-methyl aniline offered corresponding 3-aminoalkylated indoles in excellent yields.This protocol presents some remarkable features such as mild reaction conditions,simple workup procedure and excellent yields.

引用

页码：422 / 424

页数：3

共 14 条

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