ADP-RIBOSYL TRANSFERASE INHIBITORS POTENTIATING THE ANTITUMOR ACTIVITY OF PEPLOMYCIN

被引:0
|
作者
陈海英
潘启超
机构
[1] Guangzhou
[2] Research Department of Anticancer Drugs
[3] Cancer Institute
[4] Xan Yat-sen University of Medical Sciences
关键词
ADPRT; ADP-RIBOSYL TRANSFERASE INHIBITORS POTENTIATING THE ANTITUMOR ACTIVITY OF PEPLOMYCIN; PEP;
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摘要
ADP-ribosyl transferase (ADPRT)transfers the ADP-ribose portion of NAD to either chromatin protein or another ADP-ribose molecule, to form polymer of (ADP-R). This process is involved in many cellular biofunctions. In the last ten years, the evidence that ADPRT inhibitors inhibit DNA repair as well as potentiate the antitumor
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页码:236 / 240
页数:5
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