Unconventional approaches for synthesis of 2-substituted benzothiazoles

被引：0

作者：

Doraghi, Fatemeh ^{[1
]}

Edareh, Mohammad Hadi ^{[2
]}

Ghanbarlou, Mehdi ^{[1
]}

Larijani, Bagher ^{[1
]}

Mahdavi, Mohammad ^{[1
]}

机构：

[1] Univ Tehran Med Sci, Endocrinol & Metab Clin Sci Inst, Endocrinol & Metab Res Ctr, Tehran, Iran

[2] Univ Tehran, Coll Sci, Sch Chem, Tehran, Iran

来源：

ORGANIC & BIOMOLECULAR CHEMISTRY | 2025年 / 23卷 / 21期

关键词：

COPPER-CATALYZED SYNTHESIS; C-H ARYLATION; ELEMENTAL SULFUR; SUBSTITUTED BENZOTHIAZOLES; S BONDS; EFFICIENT; CYCLIZATION; DERIVATIVES; METAL; ACID;

D O I：

10.1039/d5ob00339c

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Benzothiazoles are among the most important heterocycles in pharmaceuticals, natural products, and functional materials. Hence, developing direct and sustainable routes by replacing hazardous/toxic thiol reagents with nontoxic reagents for constructing 2-substituted benzothiazoles is of utmost importance. In this review, we have highlighted many synthetic methods for the synthesis of 2-substituted benzothiazoles from different starting materials under transition metal catalysis or metal-free systems.

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页码：5046 / 5063

页数：18

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