A long march for targeted protein degradation in the new era: expanding E3 ligases

被引：0
作者：
Mi, Dazhao [1 ]
Huang, Anxin [1 ]
Song, Jingfeng [2 ,3 ]
Chen, Yihua [1 ,2 ,3 ]
机构：
[1] East China Normal Univ, Inst Biomed Sci, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China
[2] Kunming Med Univ, Sch Pharmaceut Sci, Yunnan Key Lab Pharmacol Nat Prod, Kunming 650500, Yunnan, Peoples R China
[3] Kunming Med Univ, Yunnan Coll Modern Biomed Ind, Kunming 650500, Yunnan, Peoples R China
来源：
FUTURE MEDICINAL CHEMISTRY | 2024年 / 16卷 / 21期
关键词：
E3; ligases; molecular glues; PROTACs; targeted protein degradation; undruggable therapeutic targets;
D O I：
10.1080/17568919.2024.2409618
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：2189 / 2191
页数：3
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