A short overview of dual targeting HDAC inhibitors

被引:0
作者
Liu, Wen-Bo [1 ]
Song, Jian [1 ]
Zhang, Sai-Yang [1 ,2 ]
机构
[1] Zhengzhou Univ, Sch Basic Med Sci, Zhengzhou 450001, Peoples R China
[2] State Key Lab Esophageal Canc Prevent & Treatment, Zhengzhou, Peoples R China
基金
中国国家自然科学基金;
关键词
HDACs; HDAC inhibitors; dual targeting; drug resistance; HISTONE DEACETYLASE INHIBITORS;
D O I
10.1080/17568919.2024.2437975
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:5 / 7
页数:3
相关论文
共 21 条
[11]   Designed multiple ligands. An emerging drug discovery paradigm [J].
Morphy, R ;
Rankovic, Z .
JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (21) :6523-6543
[12]   Discovery of Thieno[2,3-d]pyrimidine-Based Hydroxamic Acid Derivatives as Bromodomain-Containing Protein 4/Histone Deacetylase Dual Inhibitors Induce Autophagic Cell Death in Colorectal Carcinoma Cells [J].
Pan, Zhaoping ;
Li, Xiang ;
Wang, Yujia ;
Jiang, Qinglin ;
Jiang, Li ;
Zhang, Min ;
Zhang, Nan ;
Wu, Fengbo ;
Liu, Bo ;
He, Gu .
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (07) :3678-3700
[13]   Histone Deacetylases and Histone Deacetylase Inhibitors: Molecular Mechanisms of Action in Various Cancers [J].
Sanaei, Masumeh ;
Kavoosi, Fraidoon .
ADVANCED BIOMEDICAL RESEARCH, 2019, 8 (01) :63
[14]   Advances in targeting histone deacetylase for treatment of solid tumors [J].
Shi, Mu-Qi ;
Xu, Ying ;
Fu, Xin ;
Pan, De-Si ;
Lu, Xian-Ping ;
Xiao, Yi ;
Jiang, Yi-Zhou .
JOURNAL OF HEMATOLOGY & ONCOLOGY, 2024, 17 (01)
[15]   Development of Alkylated Hydrazides as Highly Potent and Selective Class I Histone Deacetylase Inhibitors with T cell Modulatory Properties [J].
Sun, Ping ;
Wang, Jing ;
Khan, Khadija S. ;
Yang, Weiqin ;
Ng, Billy Wai-Lung ;
Ilment, Nikita ;
Zessin, Matthes ;
Buelbuel, Emre F. ;
Robaa, Dina ;
Erdmann, Frank ;
Schmidt, Matthias ;
Romier, Christophe ;
Schutkowski, Mike ;
Cheng, Alfred Sze-Lok ;
Sippl, Wolfgang .
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (24) :16313-16337
[16]   Targeting HDAC/OAZ1 axis with a novel inhibitor effectively reverses cisplatin resistance in non-small cell lung cancer [J].
Sun, Yuhong ;
Bao, Xuefei ;
Ren, Yong ;
Jia, Lina ;
Zou, Shenglan ;
Han, Jian ;
Zhao, Mengyue ;
Han, Mei ;
Li, Hong ;
Hua, Qixiang ;
Fang, Yi ;
Yang, Jingyu ;
Wu, Chunfu ;
Chen, Guoliang ;
Wang, Lihui .
CELL DEATH & DISEASE, 2019, 10 (6)
[17]   Characterization of a novel HDAC/RXR/HtrA1 signaling axis as a novel target to overcome cisplatin resistance in human non-small cell lung cancer [J].
Wang, Wenjing ;
Zhao, Mengyue ;
Cui, Lijuan ;
Ren, Yong ;
Zhang, Jingyuan ;
Chen, Junli ;
Jia, Lina ;
Zhang, Jiayu ;
Yang, Jingyu ;
Chen, Guoliang ;
Ashby, Charles R., Jr. ;
Wu, Chunfu ;
Chen, Zhe-Sheng ;
Wang, Lihui .
MOLECULAR CANCER, 2020, 19 (01)
[18]   Perspectives on drug repurposing to overcome cancer multidrug resistance mediated by ABCB1 and ABCG2 [J].
Wu, Chung-Pu ;
Hsiao, Sung-Han ;
Wu, Yu-Shan .
DRUG RESISTANCE UPDATES, 2023, 71
[19]   Feedback Activation of Leukemia Inhibitory Factor Receptor Limits Response to Histone Deacetylase Inhibitors in Breast Cancer [J].
Zeng, Hanlin ;
Qu, Jia ;
Jin, Nan ;
Xu, Jun ;
Lin, Chenchu ;
Chen, Yi ;
Yang, Xinying ;
He, Xiang ;
Tang, Shuai ;
Lan, Xiaojing ;
Yang, Xiaotong ;
Chen, Ziqi ;
Huang, Min ;
Ding, Jian ;
Geng, Meiyu .
CANCER CELL, 2016, 30 (03) :459-473
[20]   A review of progress in o-aminobenzamide-based HDAC inhibitors with dual targeting capabilities for cancer therapy [J].
Zhang, Wei-Xin ;
Huang, Jiao ;
Tian, Xin-Yi ;
Liu, Yun-He ;
Jia, Mei-Qi ;
Wang, Wang ;
Jin, Cheng-Yun ;
Song, Jian ;
Zhang, Sai-Yang .
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 259