An improved procedure for the GMP production and formulation of the sigma-1 receptor ligand [18F]FTC146 from a precursor with a chlorine leaving group

被引：0

作者：

Maresova, A. ^{[1
]}

Cihlarova, P. ^{[1
]}

Prochazka, L. ^{[2
]}

Lebeda, O. ^{[2
]}

Popkov, A. ^{[3
,4
]}

Paul, C. ^{[5
,6
]}

Drasar, P. ^{[1
]}

Jurasek, M. ^{[1
]}

机构：

[1] Univ Chem & Technol, Prague, Czech Republic

[2] Czech Acad Sci, Husinec, Czech Republic

[3] Samo Biomed Ctr, Pardubice, Czech Republic

[4] Johannes Kepler Univ Linz, Linz, Austria

[5] Univ Hosp Bern, Bern, Switzerland

[6] Queensland Univ Technol, Brisbane, Qld, Australia

来源：

EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING | 2024年 / 51卷

关键词：

D O I：

暂无

中图分类号：

R8 [特种医学]; R445 [影像诊断学];

学科分类号：

1002 ; 100207 ; 1009 ;

摘要：

EP-0965

引用

页码：S817 / S818

页数：2

共 3 条

[1] New Positron Emission Tomography (PET) Radioligand for Imaging σ-1 Receptors in Living Subjects [J].

James, Michelle L. ;

Shen, Bin ;

Zavaleta, Cristina L. ;

Nielsen, Carsten H. ;

Mesangeau, Christophe ;

Vuppala, Pradeep K. ;

Chan, Carmel ;

Avery, Bonnie A. ;

Fishback, James A. ;

Matsumoto, Rae R. ;

Gambhir, Sanjiv S. ;

McCurdy, Christopher R. ;

Chin, Frederick T. .

JOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (19) :8272-8282

[2] A facile synthesis of precursor for the σ-1 receptor PET radioligand [18F]FTC-146 and its radiofluorination [J].

Maresova, Anna ;

Jurasek, Michal ;

Drasar, Pavel B. ;

Dolensky, Bohumil ;

Prokudina, Elena A. ;

Shalgunov, Vladimir ;

Herth, Matthias M. ;

Cumming, Paul ;

Popkov, Alexander .

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2024, 67 (02) :59-66

[3]

WALKER JM, 1990, PHARMACOL REV, V42, P355

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