Recent Advances in Design, Synthesis, and Biological Activity Studies of 1,3-Selenazoles

被引：2

作者：

Makhaeva, Nataliya A. ^{[1
]}

Amosova, Svetlana V. ^{[1
]}

Filippov, Andrey S. ^{[1
]}

Potapov, Vladimir A. ^{[1
]}

Musalov, Maxim V. ^{[1
]}

机构：

[1] Russian Acad Sci, A E Favorsky Irkutsk Inst Chem, Siberian Branch, 1 Favorsky Str, Irkutsk 664033, Russia

来源：

BIOMOLECULES | 2024年 / 14卷 / 12期

基金：

俄罗斯科学基金会;

关键词：

heterocycles; 1,3-selenazoles; synthesis; biological activity; 1,3-selenazole derivatives; ONE-POT SYNTHESIS; SELENIUM-CONTAINING HETEROCYCLES; PRIMARY SELENOCARBOXYLIC AMIDES; HIGH ANTIFUNGAL ACTIVITY; N; N-UNSUBSTITUTED SELENOUREAS; ANTIMICROBIAL EVALUATION; SELENAZOLE DERIVATIVES; EFFICIENT SYNTHESIS; HYPERVALENT IODINE; ANTIVIRAL ACTIVITY;

D O I：

10.3390/biom14121546

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

The review examines recent advances in the design and synthesis of 1,3-selenazole derivatives since 2000. Various synthetic approaches to 1,3-selenazoles and reaction conditions are discussed. The beneficial properties of 1,3-selenazoles, especially their biological activity, are emphasized. Compounds with antitumor, antiviral (HIV-1 and HIV-2), antibacterial, antifungal, antiproliferative, anticonvulsant, and antioxidant activity are highlighted.

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页数：45

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