Approaches to the Synthesis of 1,2,4-Triazolo[4,3-a]pyrimidines (Mini-Review)

被引：0

作者：

Skrylkova, A. S. ^{[1
]}

Egorov, D. M. ^{[1
,2
]}

Egorova, A. V. ^{[1
,2
]}

Manshina, A. A. ^{[3
]}

机构：

[1] St Petersburg State Inst Technol Tech Univ, St Petersburg 190013, Russia

[2] Russian Acad Sci, St Petersburg Fed Res Ctr, St Petersburg 199178, Russia

[3] St Petersburg State Univ, St Petersburg 190034, Russia

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2025年 / 95卷 / 01期

基金：

俄罗斯科学基金会;

关键词：

1,2,4-triazolo[4,3-a]pyrimidines; heterocyclic compounds; fused heterocycles; triazole; pyrimidine; cyclization; HETEROCYCLIC AMINES; DERIVATIVES; ANTIBACTERIAL; PYRIMIDINE; THIAZOLE;

D O I：

10.1134/S1070363224613322

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Abstract1,2,4-Triazolo[4,3-a]pyrimidines have significant application prospects in various fields of science, especially as biologically active compounds. This review focused on synthetic approaches of these annulated heterocyclic systems. The main trends, their development, and achievements in this field of synthesis of these classes of heterocyclic compounds, advantages and limitations of the approaches used for 1958-2024 are presented.

引用

页码：44 / 72

页数：29

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