DNA alkylation by pyrrole-imidazole seco-CBI conjugates with an indole linker: Sequence-specific DNA alkylation with 10-base-pair recognition through heterodimer formation

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Minoshima, Masafumi [1 ]
Bando, Toshikazu [1 ]
Sasaki, Shunta [1 ]
Shinohara, Ken-Ichi [1 ]
Shimizu, Tatsuhiko [1 ]
Fujimoto, Jun [1 ]
Sugiyama, Hiroshi [1 ]
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[1] Department of Chemistry, Graduate School of Science, Kyoto University, Sakyo, Kyoto 606-8502, Japan
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页码:5384 / 5390
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