Discovery of a Potent and Subtype-Selective Tyk2 Degrader Based on an Allosteric Tyk2 Inhibitor

被引：0
|
作者：
Kato, Jun-Ya [1 ]
Korenaga, Shigeru [2 ]
Iwakura, Masaru [1 ]
机构：
[1] Synthetic Research Department, ASKA Pharmaceutical Company Limited, 26-1 Muraoka-Higashi 2-Chome, Kanagawa, Fujisawa,251-8555, Japan
[2] Drug Discovery Department, ASKA Pharmaceutical Company Limited, 26-1 Muraoka-Higashi 2-Chome, Kanagawa, Fujisawa,251-8555, Japan
来源：
SSRN | 2022年
关键词：
Compilation and indexing terms; Copyright 2024 Elsevier Inc;
D O I：
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摘要：
Amino acids - Enzymes
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