Synthesis of (R)-(-)-carvone derivatives

被引:0
作者
De Sousa D.P. [1 ]
Raphael E. [2 ]
Brocksom T.J. [2 ]
机构
[1] Laboratório de Química de Produtos Naturais e Sintéticos Bioativos (LAPROBIO), Departamento de Fisiologia, Universidade Federal de Sergipe, CEP 49100-000 São Cristóvão, Sergipe
[2] Laboratório de Química Bio-Orgânica, Departamento de Química, Universidade Federal de São Carlos, 13565-905 São Carlos, SP
来源
Zeitschrift fur Naturforschung - Section B Journal of Chemical Sciences | 2010年 / 65卷 / 11期
基金
巴西圣保罗研究基金会;
关键词
Essential oils; P-Menthanes; Structure-activity relationship; Terpenes;
D O I
10.1515/znb-2010-1114
中图分类号
学科分类号
摘要
(R)-(-)-Carvone, the main constituent of spearmint oil, has several synthetic applications and is used in cosmetics, food, and pharmaceutical preparations. In a recent study we demonstrated that (R)-(-)-carvone shows significant analgesic activity. In the present report, (R)-(-)-carvone derivatives which have pharmacological potential are described. These compounds can be used in studies of structure-activity relationship to develop novel drugs. © 2010 Verlag der Zeitschrift für Naturforschung, Tübingen.
引用
收藏
页码:1381 / 1383
页数:2
相关论文
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