New regioselective synthesis of 7H-imidazo[2,1-b][1,3]thiazine and 2H,6H-pyrimido[2,1-b][1,3]thiazine derivatives

被引：0

作者：

Landreau, Cyrille ^{[1
]}

Deniaud, David ^{[1
]}

Reliquet, Alain ^{[1
]}

Meslin, Jean Claude ^{[1
]}

机构：

[1] Laboratoire de Synthese Organique, UMR CNRS 6513, Faculte des Sci. et des Techniques 2, Rue de la Houssiniere, BP 92208, 44322 Nantes Cedex 03, France

来源：

Synthesis | 2002年 / 03期

关键词：

Characterization; -; Urea;

D O I：

10.1055/s-2002-20044

中图分类号：

学科分类号：

摘要：

A series of the title compounds were prepared by the reaction of amidines 2 with α-bromoketones, acid chlorides or acrylic dienophiles. The four steps synthesis reaction from thiourea and full characterisation of 7H-imidazo[2,1-b][1,3]thiazines 4, 2H,6H-pyrimido[2,1-b][1,3]thiazin-6-ones 5, and 2H,6H-pyrimido[2,1-b][1,3]thiazines 6 are described.

引用

页码：403 / 408

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