Hypervalent iodine in synthesis 81: A one-pot procedure for the synthesis of 1H-imidazole derivatives by cyclocondensation of ketones with [Hydroxy(tosyloxy)iodo]benzene and amidines

被引：0
|
作者：
Zhang, P.-F. [1 ]
Chen, Z.-C. [1 ]
机构：
[1] Department of Chemistry, Zhejiang University (Xi-Xi Campus), Hangzhou 310028, China
来源：
Synthesis | 2001年 / 14期
关键词：
Benzene; -; Condensation; Derivatives; Ketones; Synthesis; (chemical);
D O I：
10.1055/s-2001-18059
中图分类号：
学科分类号：
摘要：
Tosyloxylation of ketones with [hydroxy(tosyloxy)iodo]benzene (HTIB), followed by treatment with amidines provides a one-pot procedure for the synthesis of 1H-imidazole derivatives with good yields.
引用
收藏
页码：2075 / 2077
相关论文
共 48 条
  • [31] "On-water" one-pot four-component synthesis of novel 1H-furo[2,3-c]pyrazole-4-amine derivatives
    Noruzian, Fatemeh
    Olyaei, Abolfazl
    Hajinasiri, Rahimeh
    RESEARCH ON CHEMICAL INTERMEDIATES, 2019, 45 (09) : 4383 - 4394
  • [32] An environmentally benign one-pot synthesis of 1,2-dihydro-1-aryl-3H-naphth[1,2-e][1,3]oxazin-3-one derivatives catalysed by phosphomolybdic acid
    Chaskar, Atul
    Vyavhare, Vimal
    Padalkar, Vikas
    Phatangare, Kiran
    Deokar, Hrushikesh
    JOURNAL OF THE SERBIAN CHEMICAL SOCIETY, 2011, 76 (01) : 21 - 26
  • [33] Efficient One-pot Synthesis, Antimicrobial and Docking Studies of Some Newer Tetrahydro-4H-benzo [1,3-e]oxazines and Related -Acylamino Ketone Derivatives
    El-Bayouki, Khairy A. M.
    Basyouni, Wahid M.
    Khatab, Tamer K.
    Kandel, Ezzat M.
    Badawy, Doria S.
    Abdel-Galil, Ebrahim
    El-Henawy, Ahmed A.
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2017, 54 (02) : 1054 - 1064
  • [34] One-Pot, Three-Component Synthesis of 3-(5-Amino-1H-pyrazol-4-yl)-3-(2-hydroxy-4,4-dimethyl-6-oxocyclohex-1-enyl)indolin-2-ones
    Ahadi, Somayeh
    Mirzaei, Peiman
    Bazgir, Ayoob
    SYNTHETIC COMMUNICATIONS, 2010, 40 (08) : 1224 - 1230
  • [35] Molecular-Iodine-Mediated, Efficient One-Pot Synthesis of 2-Iminohydantoins and 2-Amino-1H-imidazol-4(5H)-ones by Cyclodeselenization of Selenourea-Tethered Amides/Peptides
    Prabhu, Girish
    Santhosh, L.
    Nagendra, G.
    Panduranga, Veladi
    Sureshbabu, Vommina V.
    CHEMISTRYSELECT, 2017, 2 (03): : 1202 - 1206
  • [36] Base-mediated one-pot synthesis of 3,4,5,6-tetrahydro-4-substituted benzo[h] quinazoline-2(1H)-thione derivatives and evaluation of their antioxidant activity
    Sivakumar, Matam
    Prabakaran, Kaliyan
    Perumal, Muthu Seenivasa
    SYNTHETIC COMMUNICATIONS, 2018, 48 (02) : 197 - 207
  • [37] An efficient and green one-pot three-component synthesis of 4,4'-(arylmethylene) bis(1H-pyrazol5-ol) s catalyzed by 2-hydroxy ethylammonium propionate
    Zhou, Zhongqiang
    Zhang, Yuliang
    GREEN CHEMISTRY LETTERS AND REVIEWS, 2014, 7 (01) : 18 - 23
  • [38] Efficient One-Pot Synthesis of 4-Aryl-3-cyano-2,5-dihydro-1H-indeno[1,2-b]pyridin-2-one and 4-Aryl-3-cyano-1,2,5,6-tetrahydrobenzo[h]quinolin-2-one Derivatives Under Solvent-Free Conditions
    Rong, Liangce
    Han, HongXia
    Jiang, Hong
    Zhang, Qiya
    Tu, Shuajiang
    SYNTHETIC COMMUNICATIONS, 2009, 39 (06) : 1027 - 1034
  • [39] Cyclization vs. Elimination Reactions of 5-Aryl-5-hydroxy 1,3-Diones: One-Pot Synthesis of 2-Aryl-2,3-dihydro-4H-pyran-4-ones
    Khera, Rasheed Ahmad
    Ahmad, Rasheed
    Ullah, Ihsan
    Abid, Obaid-Ur-Rahman
    Fatunsin, Olumide
    Sher, Muhammad
    Villinger, Alexander
    Langer, Peter
    HELVETICA CHIMICA ACTA, 2010, 93 (09) : 1705 - 1715
  • [40] An efficient improved one-pot synthesis of thiazolo[2,3-c][1,2,4]triazol-5-yl)-2H-chromen-2-one derivatives via multi-component approach
    Penta, Santhosh
    Vedula, Rajeswar Rao
    INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 2014, 53 (01): : 115 - 119
12345