Hypervalent iodine in synthesis 81: A one-pot procedure for the synthesis of 1H-imidazole derivatives by cyclocondensation of ketones with [Hydroxy(tosyloxy)iodo]benzene and amidines

被引：0
|
作者：
Zhang, P.-F. [1 ]
Chen, Z.-C. [1 ]
机构：
[1] Department of Chemistry, Zhejiang University (Xi-Xi Campus), Hangzhou 310028, China
来源：
Synthesis | 2001年 / 14期
关键词：
Benzene; -; Condensation; Derivatives; Ketones; Synthesis; (chemical);
D O I：
10.1055/s-2001-18059
中图分类号：
学科分类号：
摘要：
Tosyloxylation of ketones with [hydroxy(tosyloxy)iodo]benzene (HTIB), followed by treatment with amidines provides a one-pot procedure for the synthesis of 1H-imidazole derivatives with good yields.
引用
收藏
页码：2075 / 2077
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