Hypervalent iodine in synthesis 81: A one-pot procedure for the synthesis of 1H-imidazole derivatives by cyclocondensation of ketones with [Hydroxy(tosyloxy)iodo]benzene and amidines

被引:0
|
作者
Zhang, P.-F. [1 ]
Chen, Z.-C. [1 ]
机构
[1] Department of Chemistry, Zhejiang University (Xi-Xi Campus), Hangzhou 310028, China
关键词
Benzene; -; Condensation; Derivatives; Ketones; Synthesis; (chemical);
D O I
10.1055/s-2001-18059
中图分类号
学科分类号
摘要
Tosyloxylation of ketones with [hydroxy(tosyloxy)iodo]benzene (HTIB), followed by treatment with amidines provides a one-pot procedure for the synthesis of 1H-imidazole derivatives with good yields.
引用
收藏
页码:2075 / 2077
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