Recent advances in the synthesis of dihydropyrimidinones via biginelli reaction

被引：1

作者：

Mushtaq, Aqsa ^{[1
]}

Munawar, Anza ^{[1
]}

Parveen, Bushra ^{[1
]}

Javed, Sadia ^{[2
]}

Zahoor, Ameer Fawad ^{[1
]}

Ali, Kulsoom Ghulam ^{[1
]}

Mansha, Asim ^{[1
]}

Irfan, Ahmad ^{[3
]}

机构：

[1] Govt Coll Univ Faisalabad, Dept Chem, Faisalabad 38000, Pakistan

[2] Govt Coll Univ Faisalabad, Dept Biochem, Faisalabad 38000, Pakistan

[3] King Khalid Univ, Dept Chem, POB 9004, Abha 61413, Saudi Arabia

来源：

JOURNAL OF THE IRANIAN CHEMICAL SOCIETY | 2024年 / 21卷 / 10期

关键词：

Biginelli reaction; Multicomponent reaction; Novel catalyst; Solvent free; ONE-POT SYNTHESIS; RECOVERABLE HETEROGENEOUS CATALYST; MICROWAVE-ASSISTED SYNTHESIS; SOLVENT-FREE; IONIC LIQUID; MULTICOMPONENT SYNTHESIS; RECYCLABLE CATALYST; ORGANIC FRAMEWORK; RAPID SYNTHESIS; SULFONIC-ACID;

D O I：

10.1007/s13738-024-03100-z

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Dihydropyrimidinone skeleton (DHMP) plays a vital part in medicinal and pharmaceutical chemistry as its derivatives exhibit a broad spectrum of anti-microbial, anti-fungal, anti-bacterial, anti-inflammatory and anti-cancer activities. Taking into account the biological significance of DHPMs, organic chemists have developed different methodologies to synthesize these biologically active target molecules. Our review focuses on the one-pot synthesis of dihydropyrimidinones via Biginelli reaction by using the efficient catalysts and reaction conditions, thereby covering the literature published since 2021.

引用

页码：2565 / 2586

页数：22

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