INCREDIBLY PRODUCTIVE ONE-POT SYNTHESIS OF QUINAZOLIN-4(3H)- ONES USING TRIS(PENTAFLUOROPHENYL)BORANE AS AN EFFECTIVE CATALYST

被引：0
作者：
Venkateswarlu, A. [1 ]
Reddy, P. Suresh [1 ]
Kumar, G. Vijay [2 ]
Krishna, M. Hari [1 ]
Thriveni, P. [1 ]
机构：
[1] Vikrama Simhapuri Univ, Dept Chem, Nellore 524320, Andhra Pradesh, India
[2] Shodana Labs, Hyderabad, India
来源：
HETEROCYCLIC LETTERS | 2024年 / 14卷 / 03期
关键词：
Quinazolin-4(3H)-ones; one-pot reaction; B(C6F5)(3); EFFICIENT SYNTHESIS; ROOM-TEMPERATURE; DERIVATIVES; ALKALOIDS;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Using isatoic anhydride, ammonium acetate, and aldehydes in DMF at mild conditions, a series of quinazolin-4(3H)-ones have been synthesized in good to exceptional yields with high selectivity in a one-pot procedure. B(C6F5)(3) effectively stimulated the reaction. Some particular benefits of the current approach are its mildness, short reaction times, and enhanced selectivity.
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页码：675 / 681
页数：7
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