共 50 条
- [1] Discovery of INCB159020, an Orally Bioavailable KRAS G12D InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (02) : 1924 - 1939Ye, Qinda论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Superstring Capital Management, New York, NY 10022 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAShvartsbart, Artem论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USALi, Zhenwu论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA SK Life Sci, King Of Prussia, PA 07652 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAGan, Pei论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Quanta Therapeut, Radnor, PA 94080 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAPolicarpo, Rocco L.论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAQi, Chao论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Synovat Therapeut, Wilmington, DE USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USARoach, Jeremy J.论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA SK Life Sci, King Of Prussia, PA 07652 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAZhu, Wenyu论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAMccammant, Matthew S.论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAHu, Bin论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USALi, Gencheng论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAYin, Haolin论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USACarlsen, Peter论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAHoang, Gia论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAZhao, Le论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USASusick, Robert论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAZhang, Fenglei论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Synovat Therapeut, Wilmington, DE USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USALai, Cheng-Tsung论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Computat Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAHassani, Abdellah Allali论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Appl Technol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAEpling, Leslie B.论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Appl Technol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAGallion, Alexandra论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Preclin Pharmacol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAKurzeja-Lipinski, Kerri论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Appl Technol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAGallagher, Karen论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Appl Technol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USARoman, Valerie论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Preclin Pharmacol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAFarren, Matthew R.论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Preclin Pharmacol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAKong, Weixi论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept DMB, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USADeller, Marc C.论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Appl Technol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAZhang, Guofeng论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Appl Technol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USACovington, Maryanne论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Appl Technol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USADiamond, Sharon论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept DMB, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAKim, Sunkyu论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Preclin Pharmacol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAYao, Wenqing论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Synovat Therapeut, Wilmington, DE USA Incyte Corp, Incyte Res Inst, Dept Preclin Pharmacol, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USASokolsky, Alexander论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USAWang, Xiaozhao论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA Incyte Corp, Incyte Res Inst, Dept Discovery Chem, Wilmington, DE 19803 USA
- [2] Discovery of SHR1127, an orally bioavailable, highly potent and selective KRAS G12D inhibitorCANCER RESEARCH, 2024, 84 (06)Li, Xin论文数: 0 引用数: 0 h-index: 0Shen, Feng论文数: 0 引用数: 0 h-index: 0Zhang, Limin论文数: 0 引用数: 0 h-index: 0Wang, Wei论文数: 0 引用数: 0 h-index: 0Kong, Luyao论文数: 0 引用数: 0 h-index: 0Bao, Yong论文数: 0 引用数: 0 h-index: 0Mao, Yuchang论文数: 0 引用数: 0 h-index: 0Wang, Zaiyong论文数: 0 引用数: 0 h-index: 0Lin, Sophie论文数: 0 引用数: 0 h-index: 0Zhang, Zhe论文数: 0 引用数: 0 h-index: 0Feng, Jun论文数: 0 引用数: 0 h-index: 0Hu, Min论文数: 0 引用数: 0 h-index: 0He, Feng论文数: 0 引用数: 0 h-index: 0
- [3] MOONRAY-01, a phase 1 study of LY3962673, a potent, orally bioavailable, and selective KRAS G12D inhibitor in KRAS G12D-mutant solid tumorsJOURNAL OF CLINICAL ONCOLOGY, 2025, 43 (4_SUPPL) : TPS845 - TPS845Lakhani, Nehal J.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAMelisi, Davide论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USASubbiah, Vivek论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAAmmakkanavar, Natraj Reddy论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAO'Reilly, Eileen M.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USACassier, Philippe Alexandre论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAWainberg, Zev A.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USADuffy, Austin G.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAPatnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAFujiwara, Yutaka论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAOberstein, Paul Eliezer论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAGarcia-Carbonero, Rocio论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAWright, Jennifer论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USALin, Aimee K.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USALi, Jian论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAAxelson, Michael D.论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USAGarrido-Laguna, Ignacio论文数: 0 引用数: 0 h-index: 0机构: START Midwest, Grand Rapids, MI USA
- [4] Preclinical characterization of LY3962673, an orally bioavailable, highly potent, and selective KRAS G12D inhibitorMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Iyer, Chandrasekar论文数: 0 引用数: 0 h-index: 0Li, Binghui论文数: 0 引用数: 0 h-index: 0Stewart, Trent R.论文数: 0 引用数: 0 h-index: 0Wang, Tao论文数: 0 引用数: 0 h-index: 0Capen, Andrew论文数: 0 引用数: 0 h-index: 0Cavitt, Rachel论文数: 0 引用数: 0 h-index: 0Anderson, Bryan D.论文数: 0 引用数: 0 h-index: 0Bocchinfuso, Wayne论文数: 0 引用数: 0 h-index: 0Zhao, Gaiying论文数: 0 引用数: 0 h-index: 0Rodriguez, Michael J.论文数: 0 引用数: 0 h-index: 0Carballares, Santiago论文数: 0 引用数: 0 h-index: 0Cooke, Andrew论文数: 0 引用数: 0 h-index: 0Bondi, Robert论文数: 0 引用数: 0 h-index: 0Burns, Lee论文数: 0 引用数: 0 h-index: 0Kelamangalath, Lakshmi论文数: 0 引用数: 0 h-index: 0Wallace, Ross论文数: 0 引用数: 0 h-index: 0Kolakowski, Gabrielle论文数: 0 引用数: 0 h-index: 0Henry, James R.论文数: 0 引用数: 0 h-index: 0Si, Chong论文数: 0 引用数: 0 h-index: 0
- [5] LY3962673, an oral, highly potent, mutant-selective, and non-covalent KRAS G12D inhibitor demonstrates robust anti-tumor activity in KRAS G12D modelsCANCER RESEARCH, 2024, 84 (06)Gong, Xueqian论文数: 0 引用数: 0 h-index: 0Gao, Hong论文数: 0 引用数: 0 h-index: 0Bender, Mark H.论文数: 0 引用数: 0 h-index: 0Ming, Wenyu论文数: 0 引用数: 0 h-index: 0Zhang, Youyan论文数: 0 引用数: 0 h-index: 0Stewart, Trent R.论文数: 0 引用数: 0 h-index: 0Yu, Chun Ping论文数: 0 引用数: 0 h-index: 0Xu, Wei Guo论文数: 0 引用数: 0 h-index: 0You, Aurthur Xintian论文数: 0 引用数: 0 h-index: 0Bian, Wen Ting论文数: 0 引用数: 0 h-index: 0Li, Binghui论文数: 0 引用数: 0 h-index: 0Wang, Tao论文数: 0 引用数: 0 h-index: 0Bian, Huimin论文数: 0 引用数: 0 h-index: 0Tandon, Manuj论文数: 0 引用数: 0 h-index: 0Capen, Andrew论文数: 0 引用数: 0 h-index: 0Cavitt, Rachel N.论文数: 0 引用数: 0 h-index: 0Anderson, Bryan D.论文数: 0 引用数: 0 h-index: 0Bocchinfuso, Wayne论文数: 0 引用数: 0 h-index: 0Klippel, Anke论文数: 0 引用数: 0 h-index: 0Iyer, Chandrasekar论文数: 0 引用数: 0 h-index: 0
- [6] Inhibition of KRAS G12D mutant with small moleculesCANCER RESEARCH, 2024, 84 (06)Lee, Dae-Hee论文数: 0 引用数: 0 h-index: 0Lee, Ji Yoon论文数: 0 引用数: 0 h-index: 0
- [7] Site-specific mutagenesis screening in KRAS G12D mutant library to uncover resistance mechanisms to KRAS G12D inhibitorsCANCER LETTERS, 2024, 591论文数: 引用数: h-index:机构:Shin, Ju-young论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Dept Integrat Biotechnol, 2066 Seobu ro, Suwon 16419, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South KoreaKim, Taeyul K.论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South KoreaKim, Kiwook论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Dept Integrat Biotechnol, 2066 Seobu ro, Suwon 16419, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South KoreaKim, Jiyun论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Dept Integrat Biotechnol, 2066 Seobu ro, Suwon 16419, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South Korea论文数: 引用数: h-index:机构:Park, Juyeong论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Grad Sch, Dept Med, Coll Med, Seoul 03722, South Korea Theragen Bio Co Ltd, Seongnam 13488, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South KoreaHan, Yoon Dae论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Dept Surg, Coll Med, Seoul 03722, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South KoreaKim, Kyung-A论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South KoreaSim, Taebo论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Severance Biomed Sci Inst, Grad Sch Med Sci, Brain Korea Project 21,Coll Med, Seoul 03722, South Korea Korea Univ, KU KIST Grad Sch Converging Sci & Technol, Seoul 02841, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South Korea论文数: 引用数: h-index:机构:Kim, Han Sang论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South Korea Yonsei Univ, Yonsei Canc Ctr, Dept Internal Med, Div Med Oncol,Coll Med, Seoul 03722, South Korea Yonsei Univ, Yonsei Canc Ctr, Div Med Oncol, Coll Med, 50 Yonsei ro, Seoul 03722, South Korea Yonsei Univ, Grad Sch Med Sci, Dept Internal Med, Brain Korea Project 21,Coll Med, Seoul 03722, South Korea
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- [9] Targeting KRAS G12D mutant tumors with the PROTAC degrader RP03707CANCER RESEARCH, 2024, 84 (06)Ji, Xiang论文数: 0 引用数: 0 h-index: 0Li, Huanping论文数: 0 引用数: 0 h-index: 0Wu, Gang论文数: 0 引用数: 0 h-index: 0Zhang, Qiguo论文数: 0 引用数: 0 h-index: 0He, Xiaolin论文数: 0 引用数: 0 h-index: 0Wu, Yanpeng论文数: 0 引用数: 0 h-index: 0Zong, Bing论文数: 0 引用数: 0 h-index: 0Xu, Xiaojin论文数: 0 引用数: 0 h-index: 0Liang, Chao论文数: 0 引用数: 0 h-index: 0Wang, Beibei论文数: 0 引用数: 0 h-index: 0Zhang, Yuwei论文数: 0 引用数: 0 h-index: 0Hu, Qingyao论文数: 0 引用数: 0 h-index: 0Zhou, Jiaxin论文数: 0 引用数: 0 h-index: 0Guo, Weihui论文数: 0 引用数: 0 h-index: 0Bai, Bing论文数: 0 引用数: 0 h-index: 0Wang, Lin论文数: 0 引用数: 0 h-index: 0Ai, Jinchao论文数: 0 引用数: 0 h-index: 0Zhang, Leduo论文数: 0 引用数: 0 h-index: 0Zhou, Honggui论文数: 0 引用数: 0 h-index: 0Sun, Shihao论文数: 0 引用数: 0 h-index: 0Wang, Yijie论文数: 0 引用数: 0 h-index: 0Wang, Youhong论文数: 0 引用数: 0 h-index: 0Fan, Qiming论文数: 0 引用数: 0 h-index: 0Chen, Dawei论文数: 0 引用数: 0 h-index: 0Zhou, Tianlun论文数: 0 引用数: 0 h-index: 0Lu, Jiasheng论文数: 0 引用数: 0 h-index: 0
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