QUANTITATIVE-ANALYSIS OF BETA-ADRENERGIC-RECEPTOR INTERACTIONS - RESOLUTION OF HIGH AND LOW AFFINITY STATES OF THE RECEPTOR BY COMPUTER MODELING OF LIGAND-BINDING DATA

被引:0
|
作者
KENT, RS
DELEAN, A
LEFKOWITZ, RJ
机构
[1] DUKE UNIV,MED CTR,DEPT BIOCHEM,DURHAM,NC 27710
[2] DUKE UNIV,MED CTR,HOWARD HUGHES MED INST LAB,DEPT MED,DIV CARDIOL,DURHAM,NC 27710
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:14 / 23
页数:10
相关论文
共 39 条
  • [1] MECHANISM OF BETA-ADRENERGIC-RECEPTOR (BAR) ACTIVATION - RESOLUTION OF HIGH AND LOW AFFINITY STATES OF THE RECEPTOR BY A COMPUTER MODELING TECHNIQUE
    KENT, RS
    DELEAN, A
    LEFKOWITZ, RJ
    CLINICAL RESEARCH, 1979, 27 (02): : A450 - A450
  • [2] ANALYSIS OF LIGAND-BINDING TO THE BETA-ADRENERGIC-RECEPTOR BY MUTAGENESIS
    STRADER, CD
    SIGAL, IS
    REGISTER, RB
    RANDS, E
    CANDELORE, M
    ZEMCIK, B
    DIXON, RAF
    FEDERATION PROCEEDINGS, 1987, 46 (06) : 2064 - 2064
  • [3] GENETIC-ANALYSIS OF LIGAND-BINDING TO THE BETA-ADRENERGIC-RECEPTOR
    DIXON, RAF
    SIGAL, IS
    REGISTER, RB
    RANDS, E
    STRADER, CD
    FEDERATION PROCEEDINGS, 1987, 46 (04) : 1444 - 1444
  • [4] BETA-ADRENERGIC-RECEPTOR LIGAND-BINDING BY RABBIT LUNG
    BLANCK, TJJ
    GILLIS, CN
    BIOCHEMICAL PHARMACOLOGY, 1979, 28 (12) : 1903 - 1909
  • [5] QUANTITATIVE-ANALYSIS OF BETA-ADRENERGIC-RECEPTOR HETEROGENEITY
    KLENEROVA, V
    HYNIE, S
    BIOMEDICA BIOCHIMICA ACTA, 1987, 46 (10) : S732 - S735
  • [6] IDENTIFICATION OF RESIDUES REQUIRED FOR LIGAND-BINDING TO THE BETA-ADRENERGIC-RECEPTOR
    STRADER, CD
    SIGAL, IS
    REGISTER, RB
    CANDELORE, MR
    RANDS, E
    DIXON, RAF
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1987, 84 (13) : 4384 - 4388
  • [7] STRUCTURAL FEATURES REQUIRED FOR LIGAND-BINDING TO THE BETA-ADRENERGIC-RECEPTOR
    DIXON, RAF
    SIGAL, IS
    CANDELORE, MR
    REGISTER, RB
    SCATTERGOOD, W
    RANDS, E
    STRADER, CD
    EMBO JOURNAL, 1987, 6 (11): : 3269 - 3275
  • [8] QUANTITATIVE RESOLUTION OF BETA-ADRENERGIC-RECEPTOR SUBTYPES BY SELECTIVE LIGAND-BINDING - APPLICATION OF A COMPUTERIZED MODEL FITTING TECHNIQUE
    HANCOCK, AA
    DELEAN, AL
    LEFKOWITZ, RJ
    MOLECULAR PHARMACOLOGY, 1979, 16 (01) : 1 - 9
  • [9] LIGAND-BINDING TO THE PORCINE ADIPOSE-TISSUE BETA-ADRENERGIC-RECEPTOR
    MERSMANN, HJ
    MCNEEL, RL
    JOURNAL OF ANIMAL SCIENCE, 1992, 70 (03) : 787 - 797
  • [10] THE BETA-ADRENERGIC-RECEPTOR - LIGAND-BINDING STUDIES ILLUMINATE THE MECHANISM OF RECEPTOR ADENYLATE-CYCLASE COUPLING
    STADEL, JM
    LEFKOWITZ, RJ
    CURRENT TOPICS IN MEMBRANES AND TRANSPORT, 1983, 18 : 45 - 66