EFFECT OF N-METHYL DEUTERATION ON ACTIVITY OF ETHYLMORPHINE N-DEMETHYLASE

被引:0
|
作者
THOMPSON, JA
HOLTZMAN, JL
机构
关键词
D O I
暂无
中图分类号
Q [生物科学];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:A914 / &
相关论文
共 50 条
  • [11] Effect of N-methyl deuteration on pharmacokinetics and pharmacodynamics of enzalutamide
    Pang, Xuchai
    Peng, Lingling
    Chen, Yuanwei
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2017, 60 (09): : 401 - 409
  • [12] Effect of N-methyl deuteration on metabolism and pharmacokinetics of enzalutamide
    Jiang, Jinfang
    Pang, Xuehai
    Li, Liang
    Dai, Xiaojian
    Diao, Xingxing
    Chen, Xiaoyan
    Zhong, Dafang
    Wang, Yingwei
    Chen, Yuanwei
    DRUG DESIGN DEVELOPMENT AND THERAPY, 2016, 10 : 2181 - 2191
  • [13] SEX-DEPENDENT DIFFERENCE IN ETHYLMORPHINE N-DEMETHYLASE IN HEPATIC MICROSOMES OF RATS
    OHMORI, S
    MORI, H
    KITAGAWA, H
    KITADA, M
    RESEARCH COMMUNICATIONS IN SUBSTANCES OF ABUSE, 1994, 15 (1-2) : 83 - 92
  • [14] RADIOMETRIC ASSAY OF ETHYLMORPHINE N-DEMETHYLASE AND O-DEETHYLASE WITH 6-H-3-ETHYLMORPHINE
    DUQUETTE, PH
    HOLTZMAN, JL
    PHARMACOLOGIST, 1977, 19 (02): : 232 - 232
  • [15] SPECIES-DIFFERENCES IN LIPID PEROXIDATION AND THEIR EFFECTS ON ETHYLMORPHINE N-DEMETHYLASE ACTIVITY IN LIVER-MICROSOMES
    KAMATAKI, T
    KITAGAWA, H
    BIOCHEMICAL PHARMACOLOGY, 1974, 23 (13) : 1915 - 1918
  • [16] EFFECT OF DRUG VEHICLES ON N-DEMETHYLASE ACTIVITY IN ISOLATED HEPATOCYTES
    SAUERS, ME
    ABRAHAM, RT
    ALVIN, JD
    ZEMAITIS, MA
    BIOCHEMICAL PHARMACOLOGY, 1980, 29 (14) : 2073 - 2076
  • [17] THE EFFECT OF NADH AND LOW OXYGEN-PRESSURE ON THE HEPATIC-MICROSOMAL ETHYLMORPHINE N-DEMETHYLASE ACTIVITY OF THE MALE-RAT
    HOLTZMAN, JL
    GANDER, JE
    ERICKSON, RR
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1983, 258 (09) : 5400 - 5404
  • [18] HEPATIC AMIDOPYRINE N-DEMETHYLASE ACTIVITY IN CALF
    FORD, EJH
    GOPINATH, C
    ADAM, SEI
    JOURNAL OF COMPARATIVE PATHOLOGY, 1972, 82 (03) : 355 - &
  • [19] EFFECTS OF ENDOGENOUS SEX-HORMONES ON MOUSE-LIVER ETHYLMORPHINE N-DEMETHYLASE
    BROWN, TR
    GREENE, FE
    ARCHIVES INTERNATIONALES DE PHARMACODYNAMIE ET DE THERAPIE, 1980, 248 (01): : 13 - 25
  • [20] DEPENDENCE OF KM AN VMAX ON SUBSTRATE CONCENTRATION FOR RAT HEPATIC MICROSOMAL ETHYLMORPHINE N-DEMETHYLASE
    HAYES, JR
    MGBODILE, MU
    CAMPBELL, TC
    BIOCHEMICAL PHARMACOLOGY, 1973, 22 (12) : 1517 - 1520