ASPARTYL ALPHA-((1-PHENYL-3-(TRIFLUOROMETHYL)PYRAZOL-5-YL)OXY)METHYL KETONES AS INTERLEUKIN-1-BETA CONVERTING-ENZYME INHIBITORS - SIGNIFICANCE OF THE P-1 AND P-3 AMIDO NITROGENS FOR ENZYME-PEPTIDE INHIBITOR BINDING

被引：49

作者：

DOLLE, RE ^{[1
]}

SINGH, J ^{[1
]}

RINKER, J ^{[1
]}

HOYER, D ^{[1
]}

PRASAD, CVC ^{[1
]}

GRAYBILL, TL ^{[1
]}

SALVINO, JM ^{[1
]}

HELASZEK, CT ^{[1
]}

MILLER, RE ^{[1
]}

ATOR, MA ^{[1
]}

机构：

[1] STERLING WINTHROP PHARMACEUT,DIV RES,DEPT BIOCHEM,COLLEGEVILLE,PA 19426

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1994年 / 37卷 / 23期

关键词：

D O I：

10.1021/jm00049a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：3863 / 3866

页数：4

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