RESEARCH ON NITROGEN AND SULFUR HETEROCYCLIC-COMPOUNDS - SYNTHESIS OF 10H-PYRROLO[1,2-A]THIENO[3,4-E][1,4]-DIAZEPIN-5(4H)-ONE AND SOME DERIVATIVES

被引：2

作者：

DAICH, A

MOREL, J

DECROIX, B

机构：

[1] Laboratoire de Chimie, UER des Sciences et des Techniques, Université du Havre, Le Havre, 76600

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1994年 / 31卷 / 02期

关键词：

D O I：

10.1002/jhet.5570310214

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of 10H-pyrrolo[1,2-a]thieno[3,4-e][1,4]diazepin-5(4H)-one (16) and some derivatives are described from methyl 3-bromomethylthiophene-4-carboxylate (5). The key step of these sequences is the intramolecular cyclization of the carbonylazides 12 and 13.

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页码：341 / 344

页数：4

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