BINDING-SITES FOR A PERIPHERAL TYPE BENZODIAZEPINE ANTAGONIST ([H-3] PK-11195) IN HUMAN IRIS

被引:12
作者
VALTIER, D
MALGOURIS, C
GILBERT, JC
GUICHENEY, P
UZAN, A
GUEREMY, C
LEFUR, G
SARAUX, H
MEYER, P
机构
[1] GRP RHONE POULENC SANTE,PHARMUKA LABS,F-92231 GENNEVILLIERS,FRANCE
[2] HOP ST ANTOINE,SERV OPHTHALMOL,F-75571 PARIS 12,FRANCE
关键词
D O I
10.1016/0028-3908(87)90146-8
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:549 / 552
页数:4
相关论文
共 50 条
  • [31] PK ('peripheral benzodiazepine') - Binding sites in the CNS indicate early and discrete brain lesions: Microautoradiographic detection of [H-3]PK11195 binding to activated microglia
    Banati, RB
    Myers, R
    Kreutzberg, GW
    JOURNAL OF NEUROCYTOLOGY, 1997, 26 (02): : 77 - 82
  • [32] CARBAMAZEPINE UP-REGULATES THE BINDING OF [H-3] PK-11195 TO PLATELETS OF EPILEPTIC PATIENTS
    WEIZMAN, A
    TANNE, Z
    KARP, L
    MARTFELD, Y
    TYANO, S
    GAVISH, M
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 141 (03) : 471 - 474
  • [33] A PERIPHERAL ANTAGONIST OF BENZODIAZEPINE RECEPTORS (PK-11195) DID NOT REVERSE BEHAVIORAL-EFFECTS OF DIAZEPAM IN MICE
    SULCOVA, A
    KRSIAK, M
    ACTIVITAS NERVOSA SUPERIOR, 1989, 31 (04): : 295 - 296
  • [34] INVIVO BINDING TO PERIPHERAL BENZODIAZEPINE BINDING-SITES IN LESIONED RAT-BRAIN - COMPARISON BETWEEN [H-3] PK11195 AND [F-18] PK14105 AS MARKERS FOR NEURONAL DAMAGE
    PRICE, GW
    AHIER, RG
    HUME, SP
    MYERS, R
    MANJIL, L
    CREMER, JE
    LUTHRA, SK
    PASCALI, C
    PIKE, V
    FRACKOWIAK, RSJ
    JOURNAL OF NEUROCHEMISTRY, 1990, 55 (01) : 175 - 185
  • [35] INTERPRETATION DU SPECTER RMN-H-3 DU PK-11195 (H-3)
    SERGENT, L
    BEAUCOURT, JP
    TETRAHEDRON LETTERS, 1985, 26 (43) : 5291 - 5292
  • [36] INCREASED DENSITIES OF BINDING-SITES FOR THE PERIPHERAL-TYPE BENZODIAZEPINE RECEPTOR-LIGAND [H-3] PK11195 IN VULNERABLE REGIONS OF THE RAT-BRAIN IN THIAMINE-DEFICIENCY ENCEPHALOPATHY
    LEONG, DK
    LE, O
    OLIVA, L
    BUTTERWORTH, RF
    JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM, 1994, 14 (01) : 100 - 105
  • [37] PK-11195, AN ANTAGONIST OF PERIPHERAL BENZODIAZEPINE RECEPTORS, REDUCES VENTRICULAR ARRHYTHMIAS DURING MYOCARDIAL ISCHEMIA AND REPERFUSION IN THE DOG
    MESTRE, M
    BOUETARD, G
    UZAN, A
    GUEREMY, C
    RENAULT, C
    DUBROEUCQ, MC
    LEFUR, G
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 112 (02) : 257 - 260
  • [38] HISTIDINE MODIFICATION WITH DIETHYLPYROCARBONATE INDUCES A DECREASE IN THE BINDING OF AN ANTAGONIST, PK-11195, BUT NOT OF AN AGONIST, RO5-4864, OF THE PERIPHERAL BENZODIAZEPINE RECEPTORS
    BENAVIDES, J
    BEGASSAT, F
    PHAN, T
    TUR, C
    UZAN, A
    RENAULT, C
    DUBROEUCQ, MC
    GUEREMY, C
    LEFUR, G
    LIFE SCIENCES, 1984, 35 (12) : 1249 - 1256
  • [39] PRESERVATION OF PERIPHERAL BENZODIAZEPINE RECEPTORS - DIFFERENTIAL-EFFECTS OF FREEZING ON [H-3] RO 5-4864 AND [H-3] PK 11195 BINDING
    BASILE, AS
    OSTROWSKI, NL
    SKOLNICK, P
    JOURNAL OF PHARMACOLOGICAL METHODS, 1987, 17 (02): : 149 - 156
  • [40] PERIPHERAL BENZODIAZEPINE BINDING-SITES - EFFECT OF PK-11195, 1-(2-CHLOROPHENYL)-N-METHYL-(1-METHYLPROPYL)-3 ISOQUINOLINECARBOXAMIDE .2. INVIVO STUDIES
    LEFUR, G
    GUILLOUX, F
    RUFAT, P
    BENAVIDES, J
    UZAN, A
    RENAULT, C
    DUBROEUCQ, MC
    GUEREMY, C
    LIFE SCIENCES, 1983, 32 (16) : 1849 - 1856