INHIBITION OF RAT PROSTATE TUMOR-GROWTH BY AN OCTAPEPTIDE ANALOG OF SOMATOSTATIN

被引:58
作者
MURPHY, WA [1 ]
LANCE, VA [1 ]
MOREAU, S [1 ]
MOREAU, JP [1 ]
COY, DH [1 ]
机构
[1] BIOMEASURE INC,HOPKINTON,MA 01748
关键词
D O I
10.1016/0024-3205(87)90073-7
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2515 / 2522
页数:8
相关论文
共 11 条
[1]  
BAUER W, 1982, LIFE SCI, V31, P1133, DOI 10.1016/0024-3205(82)90087-X
[2]  
DEQUIJADA MG, 1983, P NATL ACAD SCI-BIOL, V80, P3485
[3]   SYNTHESIS AND BIOLOGICAL-ACTIVITY OF LH-RH ANTAGONISTS MODIFIED IN POSITION-1 [J].
HORVATH, A ;
COY, DH ;
NEKOLA, MV ;
COY, EJ ;
SCHALLY, AV ;
TEPLAN, I .
PEPTIDES, 1982, 3 (06) :969-971
[4]   EFFECT OF LONG-ACTING SOMATOSTATIN-ANALOGUE, SMS 201995, ON GUT HORMONE-SECRETION IN NORMAL SUBJECTS [J].
KRAENZLIN, ME ;
WOOD, SM ;
NEUFELD, M ;
ADRIAN, TE ;
BLOOM, SR .
EXPERIENTIA, 1985, 41 (06) :738-740
[5]   STUDIES ON THE MECHANISM OF ACTION OF THE INHIBITORY EFFECT OF THE SOMATOSTATIN ANALOG SMS-201-995 ON THE GROWTH OF THE PROLACTIN ADRENOCORTICOTROPIN-SECRETING PITUITARY TUMOR-7315A [J].
LAMBERTS, SWJ ;
REUBI, JC ;
UITERLINDEN, P ;
ZUIDERWIJK, J ;
VANDENWERFF, P ;
VANHAL, P .
ENDOCRINOLOGY, 1986, 118 (06) :2188-2194
[6]   POTENT, HIGHLY SELECTIVE-INHIBITION OF GROWTH-HORMONE SECRETION BY POSITION 4 SOMATOSTATIN ANALOGS [J].
MURPHY, WA ;
MEYERS, CA ;
COY, DH .
ENDOCRINOLOGY, 1981, 109 (02) :491-495
[7]   OCTAPEPTIDE ANALOGS OF SOMATOSTATIN EXHIBITING GREATLY ENHANCED INVIVO AND INVITRO INHIBITION OF GROWTH-HORMONE SECRETION IN THE RAT [J].
MURPHY, WA ;
HEIMAN, ML ;
LANCE, VA ;
MEZO, I ;
COY, DH .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 132 (03) :922-928
[8]   THE APPLICATION OF THE PRINCIPLES OF STATISTICAL ANALYSIS TO THE BIOLOGICAL ASSAY OF HORMONES [J].
PUGSLEY, LI .
ENDOCRINOLOGY, 1946, 39 (03) :161-176
[9]   A SOMATOSTATIN ANALOG INHIBITS CHONDROSARCOMA AND INSULINOMA TUMOR-GROWTH [J].
REUBI, JC .
ACTA ENDOCRINOLOGICA, 1985, 109 (01) :108-114
[10]   SOMATOSTATIN ANALOGS - RELATIVE IMPORTANCE OF DISULFIDE BRIDGE AND OF ALA-GLY SIDE-CHAIN FOR BIOLOGICAL-ACTIVITY [J].
RIVIER, J ;
BRAZEAU, P ;
VALE, W ;
GUILLEMIN, R .
JOURNAL OF MEDICINAL CHEMISTRY, 1975, 18 (02) :123-126