HIGHLY REGIOSELECTIVE SYNTHESIS OF 1,7-DIPROTECTED 1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES

被引：35

作者：

ANELLI, PL

MURRU, M

UGGERI, F

VIRTUANI, M

机构：

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1991年 / 18期

关键词：

D O I：

10.1039/c39910001317

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Reaction of dimethylformamide diethyl acetal with monoalkylated 1,4,7,10-tetraazacyclododecane derivatives 3, followed by hydrolysis of the tricyclic intermediates 4, selectivel affords 1,7-disubstituted tetraazamacrocycles 5.

引用

页码：1317 / 1318

页数：2

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